# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA2425654 | 3 | INH | < | 50 | % | ALA2428989 | % | Homo sapiens | |||
2. | ALA2425645 | 11 | INH | < | 50 | % | ALA2428989 | % | Homo sapiens | |||
3. | ALA2425646 | 12 | INH | < | 50 | % | ALA2428989 | % | Homo sapiens | |||
4. | ALA2402081 | 37 | INH | = | -8 | % | ALA2405671 | % | Homo sapiens | |||
5. | ALA2348862 | 10b, CC214-2 | Activity | = | 96 | % | ALA2351112 | % | Homo sapiens | |||
6. | ALA2348862 | 10b, CC214-2 | Activity | = | 98 | % | ALA2352833 | % | Homo sapiens | |||
7. | ALA2348865 | 9a, CC214-1 | Activity | = | 100 | % | ALA2351112 | % | Homo sapiens | |||
8. | ALA2325940 | 42 | INH | > | 80 | % | ALA2329206 | % | Homo sapiens | |||
9. | (1S,2S,3R,4R)-3-[[5-chloro-2-[(1-ethyl-6-methoxy-2-oxo-4,5-dihydro-3H-1-benzazepin-7-yl)amino]pyrimidin-4-yl]amino]bicyclo[2.2.1]hept-5-ene-2-carboxamide | 15 | INH | < | 50 | % | ALA2044934 | % | Homo sapiens | |||
10. | (1S,2S,3R,4R)-3-[[5-chloro-2-[(1-ethyl-6-methoxy-2-oxo-4,5-dihydro-3H-1-benzazepin-7-yl)amino]pyrimidin-4-yl]amino]bicyclo[2.2.1]hept-5-ene-2-carboxamide | 15 | INH | = | 94 | % | ALA2044933 | % | Homo sapiens | |||
11. | ALA2030242 | 21 | INH | = | 89 | % | ALA2034083 | % | Homo sapiens | |||
12. | ALA1822067 | 1 | INH | = | 88 | % | ALA2034083 | % | Homo sapiens | |||
13. | ALA4098896 | 3h | Activity | = | 3.9 | % | ALA4055584 | % | Homo sapiens | |||
14. | ALA4098896 | 3h | Kd | = | 64 | nM | ALA4055574 | 7.19 | nM | Homo sapiens | ||
15. | ALA4080797 | 35 | Activity | = | 94 | % | ALA4054964 | % | Homo sapiens | |||
16. | ALA4096145 | 2 | Activity | = | 64 | % | ALA4054964 | % | Homo sapiens | |||
17. | ALA111612 | 10a | % Control | 69.6 | % | ALA4879965 | Not Active | % | Homo sapiens | |||
18. | ALA4526341 | EUB0000736 | % Control | 100 | % | ALA4879965 | Not Active | % | Homo sapiens | |||
19. | ABT-100 | EUB0000289 | % Control | 79 | % | ALA4879965 | Not Active | % | Homo sapiens | |||
20. | ALA3701197 | BDBM161028 | % Control | 100 | % | ALA4879965 | Not Active | % | Homo sapiens |