# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | N-(4-{3-[2-(methylcarbamoyl)ethyl]-5-[4'-(trifluoromethyl)-[1,1'-biphenyl]-4-yl]-1H-pyrazol-1-yl}phenyl)prop-2-ynamide | 1; Tr-87 | Activity | 0 | ALA4415383 | Active | Homo sapiens | |||||
2. | ALA3728942 | 1 | IC50 | = | 6.32 | uM | ALA3734162 | 5.20 | nM | Homo sapiens | ||
3. | ALA3732814 | 2 | IC50 | = | 50 | uM | ALA3734162 | 4.30 | nM | Homo sapiens | ||
4. | ALA3731151 | 3 | IC50 | = | 4.64 | uM | ALA3734162 | 5.33 | nM | Homo sapiens | ||
5. | ALA3728093 | 4 | IC50 | = | 24 | uM | ALA3734162 | 4.62 | nM | Homo sapiens | ||
6. | ALA3730340 | 5 | IC50 | = | 2.53 | uM | ALA3734162 | 5.60 | nM | Homo sapiens | ||
7. | ALA3730264 | 6 | IC50 | = | 16.43 | uM | ALA3734162 | 4.78 | nM | Homo sapiens | ||
8. | ALA3728456 | 7 | IC50 | = | 0.71 | uM | ALA3734162 | 6.15 | nM | Homo sapiens | ||
9. | ALA3733228 | 8 | IC50 | = | 2.01 | uM | ALA3734162 | 5.70 | nM | Homo sapiens | ||
10. | ALA3727466 | 9 | IC50 | = | 1.28 | uM | ALA3734162 | 5.89 | nM | Homo sapiens | ||
11. | ALA3727685 | 10 | IC50 | = | 4.36 | uM | ALA3734162 | 5.36 | nM | Homo sapiens | ||
12. | ALA3727376 | 11 | IC50 | = | 1.81 | uM | ALA3734162 | 5.74 | nM | Homo sapiens | ||
13. | ALA3729640 | 12 | IC50 | = | 0.741 | uM | ALA3734162 | 6.13 | nM | Homo sapiens | ||
14. | ALA3728706 | 13 | IC50 | = | 0.84 | uM | ALA3734162 | 6.08 | nM | Homo sapiens | ||
15. | ALA3730427 | 14 | IC50 | = | 7.59 | uM | ALA3734162 | 5.12 | nM | Homo sapiens | ||
16. | ALA1995927 | SID103905436 | IC50 | = | 0.009 | uM | ALA3734162 | 8.05 | nM | Homo sapiens | ||
17. | ALA3728229 | 16 | IC50 | = | 1.18 | uM | ALA3734162 | 5.93 | nM | Homo sapiens | ||
18. | ALA3728250 | 17 | IC50 | = | 0.129 | uM | ALA3734162 | 6.89 | nM | Homo sapiens | ||
19. | ALA3730512 | 18 | IC50 | = | 0.366 | uM | ALA3734162 | 6.44 | nM | Homo sapiens | ||
20. | ALA3731979 | 19 | IC50 | = | 0.32 | uM | ALA3734162 | 6.50 | nM | Homo sapiens |