# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5274306 | 15 | INH | < | 50 | % | ALA5228850 | % | Homo sapiens | |||
2. | ALA5275028 | [18F]PBR06 | Ki | = | 0.3 | nM | ALA5228264 | 9.52 | nM | Homo sapiens | ||
3. | ALA2206280 | [11C]1, [11C](R)-PK 11195 | Kd | = | 2 | nM | ALA5228262 | 8.70 | nM | Homo sapiens | ||
4. | ALA5277709 | [123I]2 | Kd | = | 10 | nM | ALA5228262 | 8.00 | nM | Homo sapiens | ||
5. | ALA286346 | Ro-54864 | Kd | = | 1.1 | nM | ALA5228258 | 8.96 | nM | Homo sapiens | ||
6. | ALA1944785 | [18F]12a, [18F]GE-180 | Ki | = | 2.4 | nM | ALA5228258 | 8.62 | nM | Homo sapiens | ||
7. | ALA54349 | Alpidem | Ki | = | 0.5 | nM | ALA5228258 | 9.30 | nM | Homo sapiens | ||
8. | ALA4066040 | 12 | % of inhibition | = | 95.5 | % | ALA5214508 | % | Homo sapiens | |||
9. | ALA5195160 | 8e | Ki | = | 71 | nM | ALA5167409 | 7.15 | nM | Homo sapiens | ||
10. | ALA5172913 | 6c | Ki | = | 271 | nM | ALA5167409 | 6.57 | nM | Homo sapiens | ||
11. | ALA5179024 | 28 | Ki | = | 108 | nM | ALA5150965 | 6.97 | nM | Homo sapiens | ||
12. | ALA5169788 | 26 | Ki | = | 202 | nM | ALA5150963 | 6.70 | nM | Homo sapiens | ||
13. | ALA5172740 | 25 | Ki | = | 438 | nM | ALA5150963 | 6.36 | nM | Homo sapiens | ||
14. | ALA5187502 | 78 | Ki | = | 3.99 | nM | ALA5141041 | 8.40 | nM | Homo sapiens | ||
15. | ALA5182943 | 107 | INH | < | 50 | % | ALA5135898 | % | Homo sapiens | |||
16. | ALA5207529 | 106 | INH | < | 50 | % | ALA5135898 | % | Homo sapiens | |||
17. | ALA5204071 | 94 | INH | < | 50 | % | ALA5135898 | % | Homo sapiens | |||
18. | ALA5170784 | 93 | INH | < | 50 | % | ALA5135898 | % | Homo sapiens | |||
19. | ALA4456416 | 22 | IC50 | = | 2.13 | nM | ALA4415150 | 8.67 | nM | Homo sapiens | ||
20. | ALA521186 | 10 | Ki | = | 0.882 | nM | ALA4415150 | 9.05 | nM | Homo sapiens |