# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA3633757 | 8k | Ki | > | 900 | nM | ALA3636767 | nM | Homo sapiens | |||
2. | ALA3634876 | 1 | Ki | = | 28.13 | nM | ALA3636924 | 7.55 | nM | Homo sapiens | ||
3. | ALA3634877 | 2 | Ki | = | 224.46 | nM | ALA3636924 | 6.65 | nM | Homo sapiens | ||
4. | ALA3634878 | 3 | Ki | = | 29.11 | nM | ALA3636924 | 7.54 | nM | Homo sapiens | ||
5. | N,N-diethyl-2-(2-(4-methoxyphenyl)-5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl)acetamide | 10, DPA-713 | Ki | = | 8.2 | nM | ALA3636924 | 8.09 | nM | Homo sapiens | ||
6. | ALA3634879 | 5 | Ki | > | 10 | uM | ALA3636924 | nM | Homo sapiens | |||
7. | ALA3634876 | 1 | Ki | = | 806 | nM | ALA3636925 | 6.09 | nM | Homo sapiens | ||
8. | ALA3634877 | 2 | Ki | = | 398.18 | nM | ALA3636925 | 6.40 | nM | Homo sapiens | ||
9. | ALA3634878 | 3 | Ki | = | 144.33 | nM | ALA3636925 | 6.84 | nM | Homo sapiens | ||
10. | N,N-diethyl-2-(2-(4-methoxyphenyl)-5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl)acetamide | 10, DPA-713 | Ki | = | 6.68 | nM | ALA3636925 | 8.18 | nM | Homo sapiens | ||
11. | ALA3634879 | 5 | Ki | > | 10 | uM | ALA3636925 | nM | Homo sapiens | |||
12. | ALA5274306 | 15 | INH | < | 50 | % | ALA5228850 | % | Homo sapiens | |||
13. | ALA5275028 | [18F]PBR06 | Ki | = | 0.3 | nM | ALA5228264 | 9.52 | nM | Homo sapiens | ||
14. | ALA2206280 | [11C]1, [11C](R)-PK 11195 | Kd | = | 2 | nM | ALA5228262 | 8.70 | nM | Homo sapiens | ||
15. | ALA5277709 | [123I]2 | Kd | = | 10 | nM | ALA5228262 | 8.00 | nM | Homo sapiens | ||
16. | ALA286346 | Ro-54864 | Kd | = | 1.1 | nM | ALA5228258 | 8.96 | nM | Homo sapiens | ||
17. | ALA1944785 | [18F]12a, [18F]GE-180 | Ki | = | 2.4 | nM | ALA5228258 | 8.62 | nM | Homo sapiens | ||
18. | ALA54349 | Alpidem | Ki | = | 0.5 | nM | ALA5228258 | 9.30 | nM | Homo sapiens | ||
19. | ALA4066040 | 12 | % of inhibition | = | 95.5 | % | ALA5214508 | % | Homo sapiens | |||
20. | ALA5195160 | 8e | Ki | = | 71 | nM | ALA5167409 | 7.15 | nM | Homo sapiens |