# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4573293 | 36 | IC50 | = | 0.7 | nM | ALA4378240 | 9.15 | nM | Mus musculus | ||
2. | (2R)-2-[5-[6-amino-5-[(1R)-1-[5-fluoro-2-(triazol-2-yl)phenyl]ethoxy]pyridin-3-yl]-4-methyl-1,3-thiazol-2-yl]propane-1,2-diol | 8e | IC50 | = | 0.8 | nM | ALA4378240 | 9.10 | nM | Mus musculus | ||
3. | ALA4436406 | 11; PF-0646392 | IC50 | = | 1.3 | nM | ALA4378240 | 8.89 | nM | Mus musculus | ||
4. | Crizotinib | 14, PF-2341066 | IC50 | = | 80 | nM | ALA4378240 | 7.10 | nM | Mus musculus | ||
5. | ALA2037208 | 4 | IC50 | = | 5.9 | uM | ALA2038865 | 5.23 | nM | Mus musculus | ||
6. | ALA2037209 | 5 | IC50 | = | 5.3 | uM | ALA2038865 | 5.28 | nM | Mus musculus | ||
7. | ALA2037220 | 16 | IC50 | = | 8.8 | uM | ALA2038865 | 5.06 | nM | Mus musculus | ||
8. | ALA2037224 | 20 | IC50 | = | 2 | uM | ALA2038865 | 5.70 | nM | Mus musculus | ||
9. | GNF 5837 | 22, GNF-5837 | IC50 | = | 3.4 | uM | ALA2038865 | 5.47 | nM | Mus musculus | ||
10. | TAE684 (NVP-TAE684) | 12, NVP-TAE684 | IC50 | < | 10 | nM | ALA1005537 | nM | Mus musculus |