| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA5285499 | KI-ARv-03 | IC50 | > | 1200 | nM | ALA5224466 | nM | Homo sapiens | |||
| 2. |  ALA5199065 | 55; KB-0742 | IC50 | > | 1200 | nM | ALA5224466 | nM | Homo sapiens | |||
| 3. |  NVP-2 | BDBM126500 | IC50 | = | 1500 | nM | ALA5224450 | 5.82 | nM | Homo sapiens | ||
| 4. |  ALA5193966 | 17a | INH | = | 91.7 | % | ALA5135744 | % | Homo sapiens | |||
| 5. |  ALA5179166 | 16a | INH | = | 97.7 | % | ALA5135744 | % | Homo sapiens | |||
| 6. |  ALA4206831 | 2; FMF-03-145-1 | Activity | = | 100 | % | ALA4185962 | % | Homo sapiens | |||
| 7. |  ALA3969370 | 19; FMF-01-086-2 | Activity | = | 99 | % | ALA4185962 | % | Homo sapiens | |||
| 8. |  ALA4174988 | 15i | Activity | = | 100 | % | ALA4157183 | % | Homo sapiens | |||
| 9. |  (5Z)-7-Oxozeaenol | 1, f152A1 | INH | = | 21.2 | % | ALA4118444 | % | Homo sapiens | |||
| 10. |  N-{2-[(5-chloro-2-{[1-(2-methoxyethyl)-1H-pyrazol-4-yl]amino}pyrimidin-4-yl)oxy]phenyl}prop-2-enamide | 25 | INH | = | 21.9 | % | ALA4118444 | % | Homo sapiens | |||
| 11. |  SM1-71 | 5 | INH | = | 3.7 | % | ALA4118444 | % | Homo sapiens | |||
| 12. |  ALA4080797 | 35 | Activity | = | 100 | % | ALA4055116 | % | Homo sapiens | |||
| 13. |  ALA4096145 | 2 | Activity | = | 95 | % | ALA4055116 | % | Homo sapiens | |||
| 14. |  ALA4092508 | 2t | Activity | = | 90 | % | ALA4044104 | % | Homo sapiens | |||
| 15. |  ALA4533018 | IM-93 | Activity | = | 99 | % | ALA4307961 | % | Homo sapiens | |||
| 16. |  JSH-150 | 40; JSH-150 | Activity | = | 32 | % | ALA4264451 | % | Homo sapiens | |||
| 17. |  PDGFRα kinase inhibitor 1 | 15i | Activity | = | 99 | % | ALA4230862 | % | Homo sapiens | |||
| 18. |  ALA4077123 | 9; CHMFL-BTK-01 | Activity | = | 100 | % | ALA4025293 | % | Homo sapiens | |||
| 19. |  BGT-226 | 53, BGT226 | Kd apparent | > | 30000 | nM | ALA3991655 | Inactive | nM | Homo sapiens | ||
| 20. |  Tideglusib | TIDEGLUSIB | Kd apparent | > | 30000 | nM | ALA3991655 | Inactive | nM | Homo sapiens |
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