# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | Dorsomorphin | 1 | IC50 | = | 68 | nM | ALA5252282 | 7.17 | nM | Homo sapiens | ||
2. | PF-06952229 | PF-06952229 | IC50 | > | 1000 | uM | ALA5224852 | nM | Homo sapiens | |||
3. | SGC GAK 1 | 15 | Kd | = | 980 | nM | ALA5213622 | 6.01 | nM | Homo sapiens | ||
4. | ML 347 | 50 | IC50 | = | 32 | nM | ALA5158315 | 7.50 | nM | Homo sapiens | ||
5. | ALA5197985 | 12e | IC50 | = | 102 | nM | ALA5133128 | 6.99 | nM | Homo sapiens | ||
6. | ALA5194265 | 12d | IC50 | = | 410 | nM | ALA5133128 | 6.39 | nM | Homo sapiens | ||
7. | ALA5190190 | 12c | IC50 | 0 | ALA5133128 | ND | Homo sapiens | |||||
8. | ALA5175201 | 12b | IC50 | = | 415 | nM | ALA5133128 | 6.38 | nM | Homo sapiens | ||
9. | ALA5196379 | 12a, racemic mixture | IC50 | > | 3000 | nM | ALA5133128 | nM | Homo sapiens | |||
10. | ALA5200241 | 11i | IC50 | = | 133 | nM | ALA5133128 | 6.88 | nM | Homo sapiens | ||
11. | ALA5178564 | 11h | IC50 | = | 762 | nM | ALA5133128 | 6.12 | nM | Homo sapiens | ||
12. | ALA5186575 | 11g | IC50 | = | 181 | nM | ALA5133128 | 6.74 | nM | Homo sapiens | ||
13. | ALA5205781 | 11f, racemic mixture | IC50 | = | 140 | nM | ALA5133128 | 6.85 | nM | Homo sapiens | ||
14. | ALA5189461 | 11e | IC50 | = | 273 | nM | ALA5133128 | 6.56 | nM | Homo sapiens | ||
15. | ALA5195236 | 11d, racemic mixture | IC50 | = | 267 | nM | ALA5133128 | 6.57 | nM | Homo sapiens | ||
16. | ALA5207070 | 11c | IC50 | = | 1202 | nM | ALA5133128 | 5.92 | nM | Homo sapiens | ||
17. | ALA5189688 | 11b | IC50 | = | 2474 | nM | ALA5133128 | 5.61 | nM | Homo sapiens | ||
18. | ALA5183080 | 11a | IC50 | = | 1083 | nM | ALA5133128 | 5.96 | nM | Homo sapiens | ||
19. | ALA5197985 | 12e | IC50 | = | 11 | nM | ALA5133124 | 7.96 | nM | Homo sapiens | ||
20. | ALA5194265 | 12d | IC50 | = | 72 | nM | ALA5133124 | 7.14 | nM | Homo sapiens |