| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA5276374 | (S)-20a; BGB-8035 | IC50 | = | 36.3 | uM | ALA5251959 | 4.44 | nM | Homo sapiens | ||
| 2. |  ALA5279102 | 21; BAY-805 | IC50 | = | 4.7 | uM | ALA5251206 | 5.33 | nM | Homo sapiens | ||
| 3. |  ALA5286594 | 615; TAK-906 | Drug metabolism | = | 43 | % | ALA5247149 | % | Homo sapiens | |||
| 4. |  BAY-091 | EUB0001564 | IC50 | = | 3.1 | uM | ALA5243038 | 5.51 | nM | Homo sapiens | ||
| 5. |  ALA5290005 | 58; BAY-297 | IC50 | = | 2.3 | uM | ALA5243038 | 5.64 | nM | Homo sapiens | ||
| 6. |  ALA5274631 | 37 | IC50 | = | 37 | uM | ALA5238208 | 4.43 | nM | Homo sapiens | ||
| 7. |  BI-3406 | I-13 | IC50 | = | 17 | uM | ALA5238208 | 4.77 | nM | Homo sapiens | ||
| 8. |  Soticlestat | SOTICLESTAT | IC50 | = | 62000 | nM | ALA5237303 | 4.21 | nM | Homo sapiens | ||
| 9. |  ALA5279363 | 58 | IC50 | > | 10 | uM | ALA5226239 | nM | Homo sapiens | |||
| 10. |  ALA5289695 | 16 | IC50 | > | 15 | uM | ALA5225641 | nM | Homo sapiens | |||
| 11. |  ALA5278512 | 4 | IC50 | = | 1.9 | uM | ALA5225582 | 5.72 | nM | Homo sapiens | ||
| 12. | ALA5278512 | 4 | INH | = | 52.6 | % | ALA5225576 | % | Homo sapiens | |||
| 13. |  ALA5291235 | 2 | INH | = | 8.5 | % | ALA5225576 | % | Homo sapiens | |||
| 14. |  ALA5290029 | 33 | IC50 | > | 40000 | uM | ALA5224658 | nM | Homo sapiens | |||
| 15. |  ALA5220884 | 49 | INH | < | 10 | % | ALA5218072 | % | Homo sapiens | |||
| 16. |  Fisogatinib (BLU-554) | BLU554 | IC50 | = | 4.7 | uM | ALA5168156 | 5.33 | nM | Homo sapiens | ||
| 17. |  N-[5-[3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-ethyl-2-oxo-1,6-naphthyridin-7-yl]-4-methoxy-2-[(1R,4R)-2-oxa-5-azabicyclo[2.2.1]heptan-5-yl]phenyl]but-2-ynamide | A34 | IC50 | = | 9.22 | uM | ALA5168156 | 5.04 | nM | Homo sapiens | ||
| 18. |  TIC10 | DORDAVIPRONE | IC50 | > | 10 | uM | ALA5167770 | nM | Homo sapiens | |||
| 19. |  ALA5191392 | 16z | IC50 | > | 10 | uM | ALA5167770 | nM | Homo sapiens | |||
| 20. |  Montelukast | 9 | IC50 | = | 0.13 | uM | ALA5167770 | 6.89 | nM | Homo sapiens |
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