# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA3122129 | 3 | IC50 | = | 0.9 | nM | ALA3124222 | 9.05 | nM | Homo sapiens | ||
2. | ALA3122128 | 2 | IC50 | = | 1.2 | nM | ALA3124222 | 8.92 | nM | Homo sapiens | ||
3. | Somatostatin-14 | 1 | IC50 | = | 1.6 | nM | ALA3124222 | 8.80 | nM | Homo sapiens | ||
4. | ALA3122127 | 1 | IC50 | = | 2.8 | nM | ALA3124222 | 8.55 | nM | Homo sapiens | ||
5. | ALA3122130 | AT2S | IC50 | = | 3.7 | nM | ALA3124222 | 8.43 | nM | Homo sapiens | ||
6. | ALA3122123 | 4 | IC50 | = | 4 | nM | ALA3124222 | 8.40 | nM | Homo sapiens | ||
7. | ALA3122124 | 5 | IC50 | = | 5.4 | nM | ALA3124222 | 8.27 | nM | Homo sapiens | ||
8. | ALA3122125 | 6 | IC50 | > | 1000 | nM | ALA3124222 | nM | Homo sapiens | |||
9. | ALA3122126 | 7 | IC50 | > | 1000 | nM | ALA3124222 | nM | Homo sapiens | |||
10. | PF 04418948 | 15, PF-04418948 | % inhibition | 0 | % | ALA4887040 | Not Active | % | Homo sapiens | |||
11. | PQCA | 4i | % inhibition | -1 | % | ALA4883044 | Not Active | % | Homo sapiens | |||
12. | BAY-899 | 36; BAY-899 | Activation (% of control) | 23 | % | ALA4884193 | % | Homo sapiens | ||||
13. | BAY-899 | 36; BAY-899 | Inhibition (% of control) | 6 | % | ALA4884168 | % | Homo sapiens | ||||
14. | ALA3480577 | DDD01251909 | Mean fold stimulation | 1.775 | ALA4883601 | Homo sapiens | ||||||
15. | PPTN | 2 | % inhibition | -5 | % | ALA4883044 | Not Active | % | Homo sapiens | |||
16. | PPTN | 2 | % inhibition | 7 | % | ALA4883044 | Not Active | % | Homo sapiens | |||
17. | PPTN | 2 | % inhibition | 17 | % | ALA4883044 | Not Active | % | Homo sapiens | |||
18. | PPTN | 2 | IC50 | 5.3 | uM | ALA4883044 | nM | Homo sapiens | ||||
19. | PPTN | 2 | % inhibition | 65 | % | ALA4883044 | Slightly Active | % | Homo sapiens | |||
20. | ALA3417525 | 69, BI665915 | % Ctrl | 146 | % | ALA4881794 | Not Active | % | Homo sapiens |