| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  A 196 | A-196 | Ki | = | 4.1 | uM | ALA5214600 | 5.39 | nM | Homo sapiens | ||
| 2. | A 196 | A-196 | % of inhibition | = | 61 | % | ALA5214599 | % | Homo sapiens | |||
| 3. |  (+)-JQ1 (DMSO solution) | (+)-JQ1 | % bound fraction | = | 48 | % | ALA5214103 | % | Homo sapiens | |||
| 4. |  ALA4562303 | MEC-B | IC50 | = | 3 | uM | ALA4396177 | 5.52 | nM | Homo sapiens | ||
| 5. | ALA4562303 | MEC-B | Ki | = | 1.6 | uM | ALA4396177 | 5.80 | nM | Homo sapiens | ||
| 6. |  ALA4579120 | 40; E40 | IC50 | = | 0.26 | uM | ALA4396177 | 6.58 | nM | Homo sapiens | ||
| 7. | ALA4579120 | 40; E40 | Ki | = | 0.14 | uM | ALA4396177 | 6.85 | nM | Homo sapiens | ||
| 8. | ALA4579120 | 40; E40 | INH | = | 98.2 | % | ALA4396151 | % | Homo sapiens | |||
| 9. |  ALA4471059 | 19 | INH | = | 49.4 | % | ALA4368590 | % | Homo sapiens | |||
| 10. |  ALA4793451 | 4j; MGS0274 | Activity | 0 | ALA4708805 | Not Active | Homo sapiens | |||||
| 11. |  ALA334014 | 3 | Activity | 0 | ALA4708805 | Not Active | Homo sapiens | |||||
| 12. |  ALA4757567 | OX0999 | INH | = | 98 | % | ALA4687886 | % | Homo sapiens | |||
| 13. |  ALA4777003 | OX1399 | INH | = | 63 | % | ALA4687886 | % | Homo sapiens | |||
| 14. |  ALA4783323 | OX1453 | INH | = | 84 | % | ALA4687886 | % | Homo sapiens | |||
| 15. |  darigabat | BDBM144227 | IC50 | = | 21 | uM | ALA4351575 | 4.68 | nM | Homo sapiens | ||
| 16. |  ALA75478 | 43 | Ki | = | 4.1 | nM | ALA4322115 | 8.39 | nM | Homo sapiens | ||
| 17. |  ALA4576324 | 24 | Ki | = | 0.4 | nM | ALA4322115 | 9.40 | nM | Homo sapiens | ||
| 18. |  CHDI 00390576 | 22 | INH | < | 25 | % | ALA4311063 | % | Homo sapiens | |||
| 19. |  ALA4437833 | 16 | INH | < | 25 | % | ALA4311063 | % | Homo sapiens | |||
| 20. |  ALA567108 | 1 | INH | = | 30 | % | ALA4309945 | % | Homo sapiens |
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