# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5306285 | EUB0002235 | delta Tm Staurosporine positive control | = | 1.138 | ALA5304832 | Homo sapiens | |||||
2. | ALA5306285 | EUB0002235 | delta Tm | = | -0.071 | ALA5304832 | Not Active | Homo sapiens | ||||
3. | ALA5308262 | EUB0002234 | delta Tm Staurosporine positive control | = | 1.138 | ALA5304728 | Homo sapiens | |||||
4. | ALA5308262 | EUB0002234 | delta Tm | = | -0.097 | ALA5304728 | Not Active | Homo sapiens | ||||
5. | ALA5308250 | EUB0002186 | delta Tm Staurosporine positive control | = | 0.178 | ALA5304631 | Homo sapiens | |||||
6. | ALA5308250 | EUB0002186 | delta Tm | = | -0.46 | ALA5304631 | Not Active | Homo sapiens | ||||
7. | ALA5306577 | EUB0002354 | delta Tm Staurosporine positive control | = | 0.178 | ALA5304532 | Homo sapiens | |||||
8. | ALA5306577 | EUB0002354 | delta Tm | = | -0.473 | ALA5304532 | Not Active | Homo sapiens | ||||
9. | BI-3812 | 44 | % Ctrl | = | 88 | % | ALA5304282 | Not Active | % | Homo sapiens | ||
10. | BI-3802 | BI-3802 | % Ctrl | = | 100 | % | ALA5304179 | Not Active | % | Homo sapiens | ||
11. | ALA3798256 | 6a | Activity | = | 91 | % | ALA3802273 | % | Homo sapiens | |||
12. | PKCθ inhibitor 14 | 14 | IC50 | > | 1000 | nM | ALA3802847 | nM | Homo sapiens | |||
13. | ALA3792850 | 26 | INH | = | -2.6 | % | ALA3794941 | % | Homo sapiens | |||
14. | ALA3793843 | 24 | INH | = | -1.8 | % | ALA3794941 | % | Homo sapiens | |||
15. | ALA508964 | 13 | INH | = | 6.9 | % | ALA3794941 | % | Homo sapiens | |||
16. | ALA3785951 | 33 | IC50 | > | 10 | uM | ALA3790001 | nM | Homo sapiens | |||
17. | ALA3786167 | 28 | IC50 | > | 10 | uM | ALA3790001 | nM | Homo sapiens | |||
18. | ALA3785500 | 3 | IC50 | > | 10 | uM | ALA3790001 | nM | Homo sapiens | |||
19. | ALA3787112 | 2 | IC50 | = | 4.8 | uM | ALA3790001 | 5.32 | nM | Homo sapiens | ||
20. | ALA3787614 | 17 | IC50 | > | 10 | uM | ALA3790001 | nM | Homo sapiens |