# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA1819577 | (S)-(aR)-22e | Activity | 0 | ALA1820476 | Active | marmosets | |||||
2. | ALA1819577 | (S)-(aR)-22e | Activity | 0 | ALA1820475 | Not Active | marmosets | |||||
3. | ALA1819577 | (S)-(aR)-22e | Activity | = | 34 | % | ALA1820474 | % | marmosets | |||
4. | BMS-846372 | 5, BMS-846372 | INH | = | 52 | % | ALA2065549 | % | marmosets | |||
5. | BMS-846372 | 5, BMS-846372 | INH | = | 52 | % | ALA2065548 | % | marmosets | |||
6. | ALA2023191 | 25c | INH | = | 31 | % | ALA2065547 | % | marmosets | |||
7. | Lapaquistat Acetate | 4a | INH | = | 25 | % | ALA2061369 | % | marmosets | |||
8. | Lapaquistat Acetate | 4a | INH | = | 29 | % | ALA2061368 | % | marmosets | |||
9. | Lapaquistat Acetate | 4a | INH | = | 14 | % | ALA2061367 | % | marmosets | |||
10. | Lapaquistat Acetate | 4a | INH | = | 23 | % | ALA2061366 | % | marmosets | |||
11. | ALA2057959 | 35f | INH | = | 12 | % | ALA2061369 | % | marmosets | |||
12. | ALA2057954 | 35a | INH | = | 16 | % | ALA2061369 | % | marmosets | |||
13. | ALA2057637 | 33b | INH | = | 24 | % | ALA2061369 | % | marmosets | |||
14. | ALA2057628 | 30b | INH | = | 21 | % | ALA2061369 | % | marmosets | |||
15. | 2-[1-[2-[(4R,6S)-8-chloro-6-(2,3-dimethoxyphenyl)-4,6-dihydropyrrolo[1,2-a][4,1]benzoxazepin-4-yl]acetyl]piperidin-4-yl]acetic acid | (4R,6S)-15a | INH | = | 28 | % | ALA2061369 | % | marmosets | |||
16. | ALA2057959 | 35f | INH | = | 21 | % | ALA2061368 | % | marmosets | |||
17. | ALA2057954 | 35a | INH | = | 52 | % | ALA2061368 | % | marmosets | |||
18. | ALA2057637 | 33b | INH | = | 21 | % | ALA2061368 | % | marmosets | |||
19. | ALA2057628 | 30b | INH | = | 23 | % | ALA2061368 | % | marmosets | |||
20. | 2-[1-[2-[(4R,6S)-8-chloro-6-(2,3-dimethoxyphenyl)-4,6-dihydropyrrolo[1,2-a][4,1]benzoxazepin-4-yl]acetyl]piperidin-4-yl]acetic acid | (4R,6S)-15a | INH | = | 9 | % | ALA2061368 | % | marmosets |