# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | Remibrutinib (LOU064) | 25; LOU064 | Activity | 0 | ALA4358617 | Not Active | Homo sapiens | |||||
2. | Belzutifan | 2; PT2977 | Activity | 0 | ALA4312716 | Not Active | Homo sapiens | |||||
3. | ALA4202767 | 56 | Activity | <= | 25 | % | ALA4187098 | % | Homo sapiens | |||
4. | PQCA | 4i | % inhibition | 2 | % | ALA4883026 | Not Active | % | Homo sapiens | |||
5. | ALA3480577 | DDD01251909 | Mean fold stimulation | 0.825 | ALA4883380 | Homo sapiens | ||||||
6. | PPTN | 2 | % inhibition | 19 | % | ALA4883026 | Not Active | % | Homo sapiens | |||
7. | ABT 724 | 3a | % inhibition | < | 10 | % | ALA4880349 | Not Active | % | Homo sapiens | ||
8. | ABT-100 | EUB0000289 | % inhibition | < | 10 | % | ALA4880187 | Not Active | % | Homo sapiens | ||
9. | ALA3697701 | BDBM161012 | % inhibition | 5 | % | ALA4880130 | Not Active | % | Homo sapiens | |||
10. | ALA3926775 | 1 | IC50 | = | 2700 | nM | ALA3880098 | 5.57 | nM | Homo sapiens | ||
11. | ALA3956728 | 2 | IC50 | = | 1000 | nM | ALA3880098 | 6.00 | nM | Homo sapiens | ||
12. | ALA3966583 | 3 | IC50 | = | 8000 | nM | ALA3880098 | 5.10 | nM | Homo sapiens | ||
13. | ALA3961540 | 4 | IC50 | = | 1000 | nM | ALA3880098 | 6.00 | nM | Homo sapiens | ||
14. | ALA3913089 | 5 | IC50 | = | 2700 | nM | ALA3880098 | 5.57 | nM | Homo sapiens | ||
15. | ALA3910434 | 6 | IC50 | = | 1300 | nM | ALA3880098 | 5.89 | nM | Homo sapiens | ||
16. | ALA3979946 | 7; 15 | IC50 | = | 910 | nM | ALA3880098 | 6.04 | nM | Homo sapiens | ||
17. | ALA3977579 | 8 | IC50 | = | 1000 | nM | ALA3880098 | 6.00 | nM | Homo sapiens | ||
18. | ALA3934499 | 9 | IC50 | = | 890 | nM | ALA3880098 | 6.05 | nM | Homo sapiens | ||
19. | dithiipin-1,1,4,4-tetroxide analogue 7 | 10 | IC50 | = | 190 | nM | ALA3880098 | 6.72 | nM | Homo sapiens | ||
20. | ALA3932833 | 11 | IC50 | = | 600 | nM | ALA3880098 | 6.22 | nM | Homo sapiens |