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# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | Adefovir | 2 | Km | = | 6 | mM | ALA3378152 | nM | Homo sapiens | |||
2. | Tenofovir | 1 | Km | = | 3 | mM | ALA3378152 | nM | Homo sapiens | |||
3. | ALA3322196 | 8 | Km | = | 0.42 | mM | ALA3378152 | nM | Homo sapiens | |||
4. | ALA3322195 | 5 | Km | 0 | ALA3378152 | Not Active | Homo sapiens | |||||
5. | 2′-Deoxyadenosine 5′-monophosphate | SID8139940 | Km | = | 0.21 | mM | ALA3378152 | nM | Homo sapiens | |||
6. | 5'-Adenylic Acid | AMPs from Table 3 | Km | = | 0.38 | mM | ALA3378152 | nM | Homo sapiens | |||
7. | Adefovir | 2 | Kcat/Km | = | 250 | 10'6/M/s | ALA3378154 | 10'6/M/s | Homo sapiens | |||
8. | Tenofovir | 1 | Kcat/Km | = | 800 | 10'6/M/s | ALA3378154 | 10'6/M/s | Homo sapiens | |||
9. | ALA3322196 | 8 | Kcat/Km | = | 0.025 | 10'6/M/s | ALA3378154 | 10'6/M/s | Homo sapiens | |||
10. | ALA3322195 | 5 | Kcat/Km | 0 | ALA3378154 | Not Active | Homo sapiens | |||||
11. | 2′-Deoxyadenosine 5′-monophosphate | SID8139940 | Kcat/Km | = | 0.5 | 10'6/M/s | ALA3378154 | 10'6/M/s | Homo sapiens | |||
12. | 5'-Adenylic Acid | AMPs from Table 3 | Kcat/Km | = | 0.21 | 10'6/M/s | ALA3378154 | 10'6/M/s | Homo sapiens | |||
13. | 5'-Adenylic Acid | AMPs from Table 3 | Kcat | = | 80 | /s | ALA3378152 | /s | Homo sapiens | |||
14. | 2′-Deoxyadenosine 5′-monophosphate | SID8139940 | Kcat | = | 110 | /s | ALA3378152 | /s | Homo sapiens | |||
15. | ALA3322195 | 5 | Kcat | 0 | ALA3378152 | Not Active | Homo sapiens | |||||
16. | ALA3322196 | 8 | Kcat | = | 1.06 | /s | ALA3378152 | /s | Homo sapiens | |||
17. | Tenofovir | 1 | Kcat | = | 2.4 | /s | ALA3378152 | /s | Homo sapiens | |||
18. | Adefovir | 2 | Kcat | = | 1.5 | /s | ALA3378152 | /s | Homo sapiens | |||
19. | PF-562271 | PF-562271 | Kd apparent | > | 30000 | nM | ALA3991622 | Inactive | nM | Homo sapiens | ||
20. | RAF265 (CHIR-265) | CHIR-265/RAF-265 | Kd apparent | > | 30000 | nM | ALA3991622 | Inactive | nM | Homo sapiens |
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