# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | BTZO 1 | EUB0000301 | Kd | = | 68.6 | nM | ALA5210492 | 7.16 | nM | Homo sapiens | ||
2. | ALA4561806 | EUB0001135 | MEC1.5 | > | 1000 | nM | ALA5210037 | nM | Homo sapiens | |||
3. | BTZO 1 | EUB0000301 | MEC1.5 | = | 16 | nM | ALA5210033 | nM | Homo sapiens | |||
4. | ALA5203854 | 4-MPP | Kcat/Km | = | 0.98 | 10^4/M/s | ALA5157689 | 10^4/M/s | Homo sapiens | |||
5. | ALA5174816 | 4-HPP | Kcat/Km | = | 2.6 | 10^4/M/s | ALA5157689 | 10^4/M/s | Homo sapiens | |||
6. | ALA5197757 | 4-CPP | Kcat/Km | = | 4.3 | 10^4/M/s | ALA5157689 | 10^4/M/s | Homo sapiens | |||
7. | ALA5185683 | PP | Kcat/Km | = | 1.9 | 10^4/M/s | ALA5157689 | 10^4/M/s | Homo sapiens | |||
8. | ALA5185683 | PP | Kcat | = | 14 | /s | ALA5157681 | /s | Homo sapiens | |||
9. | ALA5197757 | 4-CPP | Kcat | = | 25 | /s | ALA5157681 | /s | Homo sapiens | |||
10. | ALA5174816 | 4-HPP | Kcat | = | 25 | /s | ALA5157681 | /s | Homo sapiens | |||
11. | ALA5203854 | 4-MPP | Kcat | = | 13 | /s | ALA5157681 | /s | Homo sapiens | |||
12. | ALA5185683 | PP | Km | = | 0.76 | mM | ALA5157678 | nM | Homo sapiens | |||
13. | ALA5197757 | 4-CPP | Km | = | 0.6 | mM | ALA5157678 | nM | Homo sapiens | |||
14. | ALA5174816 | 4-HPP | Km | = | 0.94 | mM | ALA5157678 | nM | Homo sapiens | |||
15. | ALA5203854 | 4-MPP | Km | = | 1.3 | mM | ALA5157678 | nM | Homo sapiens | |||
16. | (+)-Nebivolol | Nebivolol | INH | 0 | ALA5133036 | Active | % | Homo sapiens | ||||
17. | 6,7-Dihydroxycoumarin | 18 | INH | 0 | ALA5133036 | Active | % | Homo sapiens | ||||
18. | Esculin hydrate | 7 | INH | 0 | ALA5133036 | Active | % | Homo sapiens | ||||
19. | metaraminol | Metaraminol | INH | 0 | ALA5133036 | Active | % | Homo sapiens | ||||
20. | Histamine, Free Base | histamine | INH | 0 | ALA5133036 | Active | % | Homo sapiens |