# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA2152768 | 3 | INH | = | 1.2 | % | ALA2157432 | % | Homo sapiens | |||
2. | CCT128930 | 25 | INH | = | 0 | % | ALA3134934 | % | Homo sapiens | |||
3. | ALA598194 | 21, CCT129524 | INH | = | 5.5 | % | ALA3136705 | % | Homo sapiens | |||
4. | 4-(1H-Purin-6-yl)morpholine | Table S1, R3C1 | INH | = | 46 | % | ALA3136991 | % | Homo sapiens | |||
5. | ALA560373 | 10 | INH | = | 0 | % | ALA3135456 | % | Homo sapiens | |||
6. | ALA1928677 | 8 | INH | = | 22 | % | ALA3136354 | % | Homo sapiens | |||
7. | ALA1928692 | 23 | INH | = | 0 | % | ALA3136641 | % | Homo sapiens | |||
8. | SAR-020106 | (R)-3, SAR-020106 | INH | = | 19 | % | ALA3135069 | % | Homo sapiens | |||
9. | 7-Azaindole | 7-Azaindole (table 1) | INH | = | 31.5 | % | ALA3136793 | % | Homo sapiens | |||
10. | Borussertib | EUB0000645a | % Inhibition | -1 | % | ALA4888224 | Not Active | % | Homo sapiens | |||
11. | BAY-091 | EUB0001564 | % inhibition | -2.41 | % | ALA4888022 | Not Active | % | Homo sapiens | |||
12. | BI 605906 | BI605906 | % Ctrl | 112 | % | ALA4887564 | Not Active | % | Homo sapiens | |||
13. | Defactinib | DEFACTINIB | % inhibition | 10 | % | ALA4887143 | Not Active | % | Homo sapiens | |||
14. | ALA2180408 | Figure 27, R1C1 | % inhibition | 5 | % | ALA4886333 | Not Active | % | Homo sapiens | |||
15. | ALA4475494 | 19 | % Inhibition | 6 | % | ALA4886063 | Not Active | % | Homo sapiens | |||
16. | ALA4097778 | 16h | pIC50 | 6 | ALA4885408 | nM | Homo sapiens | |||||
17. | ALA4549667 | EUB0000720 | pIC50 | 6 | ALA4885122 | nM | Homo sapiens | |||||
18. | ALA4088216 | 14 | pIC50 | 6 | ALA4884831 | nM | Homo sapiens | |||||
19. | ALA4580220 | EUB0000311 | % residual kinase activity | 99 | % | ALA4884448 | Not Active | % | Homo sapiens | |||
20. | Skepinone-L | 2, Skepinone-L | % Residual activity with Skepinone-L | 109 | % | ALA4884066 | Not Active | % | Homo sapiens |