# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | Sotrastaurin | 1 | INH | = | 80 | % | ALA5159035 | % | Homo sapiens | |||
2. | ALA5206391 | 2l | INH | = | 2 | % | ALA5158992 | % | Homo sapiens | |||
3. | ALA5170735 | 2k | INH | = | 6 | % | ALA5158992 | % | Homo sapiens | |||
4. | ALA5198734 | 2j | INH | = | 6 | % | ALA5158992 | % | Homo sapiens | |||
5. | ALA5185816 | 2i | INH | = | 9 | % | ALA5158992 | % | Homo sapiens | |||
6. | ALA5188904 | 2h | INH | = | 7 | % | ALA5158992 | % | Homo sapiens | |||
7. | ALA5189743 | 2g | INH | = | 3 | % | ALA5158992 | % | Homo sapiens | |||
8. | ALA5187518 | 2f | INH | = | 4 | % | ALA5158992 | % | Homo sapiens | |||
9. | ALA5200234 | 2e | INH | = | 12 | % | ALA5158992 | % | Homo sapiens | |||
10. | ALA5204938 | 2d | INH | = | 7 | % | ALA5158992 | % | Homo sapiens | |||
11. | ALA5197769 | 2c | INH | = | 7 | % | ALA5158992 | % | Homo sapiens | |||
12. | ALA5186128 | 2b | INH | = | 9 | % | ALA5158992 | % | Homo sapiens | |||
13. | ALA5185043 | 2a | INH | = | 9 | % | ALA5158992 | % | Homo sapiens | |||
14. | ALA4644763 | 21 | IC50 | = | 0.013 | uM | ALA5127341 | 7.89 | nM | Homo sapiens | ||
15. | ALA4637961 | 6 | IC50 | = | 26 | uM | ALA5127341 | 4.58 | nM | Homo sapiens | ||
16. | ALA4645167 | 8 | IC50 | = | 14 | uM | ALA5127341 | 4.85 | nM | Homo sapiens | ||
17. | ALA4635482 | 37 | IC50 | = | 0 | uM | ALA5127341 | 10.00 | nM | Homo sapiens | ||
18. | ALA4633862 | 7 | IC50 | = | 60 | uM | ALA5127341 | 4.22 | nM | Homo sapiens | ||
19. | ALA4633319 | 9 | IC50 | = | 2 | uM | ALA5127341 | 5.70 | nM | Homo sapiens | ||
20. | JTE-952 | JTE-952; (S)-8b | IC50 | > | 1000 | nM | ALA4424906 | nM | Homo sapiens |