# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA3088243 | [18F]11, [18F]FIMX | Stability | = | 98.9 | % | ALA3089869 | % | Macaca mulatta | |||
2. | ALA3088243 | [18F]11, [18F]FIMX | Fu | = | 0.012 | ALA3089868 | Macaca mulatta | |||||
3. | ALA3088243 | [18F]11, [18F]FIMX | Drug uptake | = | 43 | % | ALA3089865 | % | Macaca mulatta | |||
4. | ALA3088243 | [18F]11, [18F]FIMX | Drug uptake | = | 31 | % | ALA3089864 | % | Macaca mulatta | |||
5. | ALA3088243 | [18F]11, [18F]FIMX | Drug uptake | 0 | ALA3089863 | Active | Macaca mulatta | |||||
6. | ALA3088243 | [18F]11, [18F]FIMX | Drug uptake | = | 19 | % | ALA3089862 | % | Macaca mulatta | |||
7. | ALA3088243 | [18F]11, [18F]FIMX | Drug uptake | = | 23 | % | ALA3089861 | % | Macaca mulatta | |||
8. | ALA3088243 | [18F]11, [18F]FIMX | Drug uptake | = | 10 | % | ALA3089860 | % | Macaca mulatta | |||
9. | ALA3088243 | [18F]11, [18F]FIMX | Drug uptake | = | 1 | % | ALA3089859 | % | Macaca mulatta | |||
10. | ALA3088243 | [18F]11, [18F]FIMX | Drug uptake | = | 21 | % | ALA3089858 | % | Macaca mulatta | |||
11. | ALA3088243 | [18F]11, [18F]FIMX | Drug uptake | = | 26 | % | ALA3089857 | % | Macaca mulatta | |||
12. | ALA2441636 | 5a(SS), SAR110068 | Stability | 0 | ALA2443802 | Stable | % | Macaca mulatta | ||||
13. | ALA2441952 | 2s, BMS-767778, More active atropisomer | PPB | = | 16 | % | ALA2444164 | % | Macaca mulatta | |||
14. | MK-0974 | 38, MK-0974 | Fu | = | 3.8 | % | ALA2434390 | Macaca mulatta | ||||
15. | MK-3207 | 3, MK-3207 | Fu | = | 9.6 | % | ALA2434390 | Macaca mulatta | ||||
16. | ALA2431254 | 3 | Fu | = | 42.9 | % | ALA2434390 | Macaca mulatta | ||||
17. | ALA2431255 | 4 | Fu | = | 33.3 | % | ALA2434390 | Macaca mulatta | ||||
18. | ALA2431256 | 5 | Fu | = | 20.5 | % | ALA2434390 | Macaca mulatta | ||||
19. | ALA2431247 | 6 | Fu | = | 11.7 | % | ALA2434390 | Macaca mulatta | ||||
20. | ALA2035981 | 4 | Fu | = | 10.4 | % | ALA2434390 | Macaca mulatta |