# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5206366 | 13; JNJ-64264681 | IC50 | = | 0.089 | uM | ALA5152661 | 7.05 | nM | Homo sapiens | ||
2. | ALA4851021 | 27 | IC50 | = | 0.084 | uM | ALA5152661 | 7.08 | nM | Homo sapiens | ||
3. | ALA5195095 | 2 | IC50 | = | 1.2 | nM | ALA5128304 | 8.92 | nM | Homo sapiens | ||
4. | ALA4448056 | 23e | pIC50 | = | 7.9 | ALA4404021 | 7.90 | nM | Homo sapiens | |||
5. | ALA4438171 | 24; I-BET469 | pIC50 | = | 7.6 | ALA4404021 | 7.60 | nM | Homo sapiens | |||
6. | ALA4456922 | 20a | pIC50 | = | 6.6 | ALA4404021 | 6.60 | nM | Homo sapiens | |||
7. | ALA4438171 | 24; I-BET469 | pIC50 | = | 7.7 | ALA4404020 | 7.70 | nM | Homo sapiens | |||
8. | ALA4456922 | 20a | pIC50 | = | 6.7 | ALA4404020 | 6.70 | nM | Homo sapiens | |||
9. | SB 203580 (DMSO solution) | 9 | IC50 | = | 3202 | nM | ALA4395857 | 5.50 | nM | Homo sapiens | ||
10. | ALA4536012 | 20c | IC50 | = | 317 | nM | ALA4395857 | 6.50 | nM | Homo sapiens | ||
11. | ALA4474903 | 1c | IC50 | = | 541 | nM | ALA4395857 | 6.27 | nM | Homo sapiens | ||
12. | AZD9898 | BDBM223287 | Activity | 0 | ALA4378221 | Dose-dependent effect | Homo sapiens | |||||
13. | AZD9898 | BDBM223287 | Activity | 0 | ALA4378220 | Dose-dependent effect | Homo sapiens | |||||
14. | AZD9898 | BDBM223287 | Activity | 0 | ALA4378219 | Dose-dependent effect | Homo sapiens | |||||
15. | AZD9898 | BDBM223287 | Activity | 0 | ALA4378218 | Dose-dependent effect | Homo sapiens | |||||
16. | ALA4862372 | 36; GSK097 | pIC50 | = | 6.8 | ALA4809912 | 6.80 | nM | Homo sapiens | |||
17. | ALA4867556 | 43 | pIC50 | = | 6.9 | ALA4809912 | 6.90 | nM | Homo sapiens | |||
18. | ALA4857098 | 40 | pIC50 | = | 6.5 | ALA4809912 | 6.50 | nM | Homo sapiens | |||
19. | ALA4868170 | 39 | pIC50 | = | 6.6 | ALA4809912 | 6.60 | nM | Homo sapiens | |||
20. | ALA4873182 | 32 | pIC50 | = | 7 | ALA4809912 | 7.00 | nM | Homo sapiens |