# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | I-BET762 | I-BET, GSK525762A | Fu | = | 0.19 | ALA2433585 | Homo sapiens | |||||
2. | ALA2425240 | 4a | t1/2 | = | 38 | min | ALA2429464 | hr | Homo sapiens | |||
3. | ALA2425241 | 4b | t1/2 | = | 62 | min | ALA2429460 | hr | Homo sapiens | |||
4. | ALA2425242 | 4c | t1/2 | = | 94 | min | ALA2429456 | hr | Homo sapiens | |||
5. | ALA2402509 | 44 | IC50 | = | 55 | nM | ALA2405800 | 7.26 | nM | Homo sapiens | ||
6. | ALA2087747 | 45 | IC50 | = | 124 | nM | ALA2092447 | 6.91 | nM | Homo sapiens | ||
7. | ALA2087746 | 44 | IC50 | = | 822 | nM | ALA2092447 | 6.08 | nM | Homo sapiens | ||
8. | ALA2087745 | 43 | IC50 | > | 5000 | nM | ALA2092447 | nM | Homo sapiens | |||
9. | ALA2087744 | 42 | IC50 | = | 1466 | nM | ALA2092447 | 5.83 | nM | Homo sapiens | ||
10. | ALA2087743 | 41 | IC50 | = | 467 | nM | ALA2092447 | 6.33 | nM | Homo sapiens | ||
11. | AL 8697 | 40 | IC50 | = | 116 | nM | ALA2092447 | 6.94 | nM | Homo sapiens | ||
12. | ALA2087741 | 39 | IC50 | = | 516 | nM | ALA2092447 | 6.29 | nM | Homo sapiens | ||
13. | ALA2087526 | 31 | IC50 | = | 105 | nM | ALA2092447 | 6.98 | nM | Homo sapiens | ||
14. | ALA2087525 | 30 | IC50 | = | 1110 | nM | ALA2092447 | 5.96 | nM | Homo sapiens | ||
15. | ALA2087524 | 29 | IC50 | = | 84 | nM | ALA2092447 | 7.08 | nM | Homo sapiens | ||
16. | ALA2087522 | 27 | IC50 | = | 278 | nM | ALA2092447 | 6.56 | nM | Homo sapiens | ||
17. | ALA2087521 | 26 | IC50 | = | 177 | nM | ALA2092447 | 6.75 | nM | Homo sapiens | ||
18. | ALA2087520 | 25 | IC50 | = | 1839 | nM | ALA2092447 | 5.74 | nM | Homo sapiens | ||
19. | ALA2087517 | 22 | IC50 | = | 257 | nM | ALA2092447 | 6.59 | nM | Homo sapiens | ||
20. | ALA2087516 | 21 | IC50 | = | 1056 | nM | ALA2092447 | 5.98 | nM | Homo sapiens |