# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA3087669 | 3h | Drug metabolism | < | 5 | % | ALA3089240 | % | Oryctolagus cuniculus | |||
2. | ALA2441636 | 5a(SS), SAR110068 | Stability | 0 | ALA2443800 | Stable | % | Oryctolagus cuniculus | ||||
3. | ALA2419745 | LB30870 | 2aPTT | = | 1.1 | uM | ALA2423869 | uM | Oryctolagus cuniculus | |||
4. | ALA2419745 | LB30870 | 2PT | = | 2.04 | uM | ALA2423867 | uM | Oryctolagus cuniculus | |||
5. | ALA2419745 | LB30870 | 2TT | = | 0.019 | uM | ALA2423861 | uM | Oryctolagus cuniculus | |||
6. | ALA2419745 | LB30870 | Activity | 0 | ALA2423869 | Dose-dependent effect | Oryctolagus cuniculus | |||||
7. | ALA2419745 | LB30870 | Activity | 0 | ALA2423867 | Dose-dependent effect | Oryctolagus cuniculus | |||||
8. | ALA2419745 | LB30870 | Activity | 0 | ALA2423861 | Dose-dependent effect | Oryctolagus cuniculus | |||||
9. | zavegepant | 3, BMS-742413 | Cp | > | 10 | nM | ALA2400606 | nM | Oryctolagus cuniculus | |||
10. | ALA2381898 | 2l | Cp | = | 5 | uM | ALA2384220 | uM | Oryctolagus cuniculus | |||
11. | ALA2312933 | A | Cp(f)ss | = | 0.8 | uM | ALA2319029 | uM | Oryctolagus cuniculus | |||
12. | ALA2313230 | 2f | Cp(f)ss | = | 0.6 | uM | ALA2319029 | uM | Oryctolagus cuniculus | |||
13. | Scutellarin | Scutellarin | TT | = | 21.35 | s | ALA2317878 | s | Oryctolagus cuniculus | |||
14. | scutellarein-7-O-glucoside | 3a | TT | = | 18.13 | s | ALA2317878 | s | Oryctolagus cuniculus | |||
15. | ALA2312738 | 3b | TT | = | 20.54 | s | ALA2317878 | s | Oryctolagus cuniculus | |||
16. | ALA2312737 | 3c | TT | = | 29.17 | s | ALA2317878 | s | Oryctolagus cuniculus | |||
17. | Scutellarin | Scutellarin | PT | = | 6.91 | s | ALA2317877 | s | Oryctolagus cuniculus | |||
18. | scutellarein-7-O-glucoside | 3a | PT | = | 7.81 | s | ALA2317877 | s | Oryctolagus cuniculus | |||
19. | ALA2312738 | 3b | PT | = | 6.57 | s | ALA2317877 | s | Oryctolagus cuniculus | |||
20. | ALA2312737 | 3c | PT | = | 9.93 | s | ALA2317877 | s | Oryctolagus cuniculus |