# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | VU0404251 | 8v, VU0404251 | Drug uptake | = | 7.4 | uM | ALA2156683 | uM | Rattus norvegicus | |||
2. | VU0404251 | 8v, VU0404251 | Tmax | = | 30 | min | ALA2156681 | hr | Rattus norvegicus | |||
3. | VU0404251 | 8v, VU0404251 | Cmax | = | 435 | nM | ALA2156680 | nM | Rattus norvegicus | |||
4. | VU0404251 | 8v, VU0404251 | Ratio AUC | = | 0.05 | ALA2156679 | Rattus norvegicus | |||||
5. | VU0404251 | 8v, VU0404251 | AUC | = | 1.2 | uM.hr | ALA2156678 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | Rattus norvegicus | ||
6. | VU0404251 | 8v, VU0404251 | Fu | = | 1 | % | ALA2156672 | Rattus norvegicus | ||||
7. | ALA2152121 | 27o | Drug uptake | = | 126 | ng/g | ALA2156966 | ng/g | Rattus norvegicus | |||
8. | ALA2152121 | 27o | Drug uptake | = | 441 | ng/g | ALA2156963 | ng/g | Rattus norvegicus | |||
9. | ALA2152121 | 27o | Drug uptake | = | 538 | ng/g | ALA2156960 | ng/g | Rattus norvegicus | |||
10. | ALA2152120 | 27n | Drug uptake | = | 485 | ng/g | ALA2156965 | ng/g | Rattus norvegicus | |||
11. | ALA2152120 | 27n | Drug uptake | = | 1220 | ng/g | ALA2156962 | ng/g | Rattus norvegicus | |||
12. | ALA2152120 | 27n | Drug uptake | = | 1004 | ng/g | ALA2156959 | ng/g | Rattus norvegicus | |||
13. | ALA2151638 | 17c | Drug uptake | = | 84 | ng/g | ALA2157276 | ng/g | Rattus norvegicus | |||
14. | ALA2151497 | 13n | Drug uptake | = | 280 | ng/g | ALA2157276 | ng/g | Rattus norvegicus | |||
15. | ALA2152119 | 27m | Drug uptake | = | 843 | ng/g | ALA2156965 | ng/g | Rattus norvegicus | |||
16. | ALA2152119 | 27m | Drug uptake | = | 1042 | ng/g | ALA2156962 | ng/g | Rattus norvegicus | |||
17. | ALA2152119 | 27m | Drug uptake | = | 932 | ng/g | ALA2156959 | ng/g | Rattus norvegicus | |||
18. | PF-04995274 | 1 | AUC | = | 1790 | ng.hr/g | ALA2154192 | ng.hr/g | Rattus norvegicus | |||
19. | ALA520648 | 29 | Occ50 | = | 0.2 | uM | ALA2149628 | uM | Rattus norvegicus | |||
20. | ALA2147529 | 5 | Drug uptake | 0 | ALA2149949 | Not Active | Rattus norvegicus |