# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA1761321 | 31 | Drug uptake | = | 2.1 | uM | ALA2396035 | uM | Rattus norvegicus | |||
2. | ALA1761313 | 22 | Drug uptake | = | 5.1 | uM | ALA2396035 | uM | Rattus norvegicus | |||
3. | ALA2391969 | 5 | Drug uptake | = | 4.4 | uM | ALA2396035 | uM | Rattus norvegicus | |||
4. | ALA373257 | 11 | Drug uptake | = | 0.2 | uM | ALA2396035 | uM | Rattus norvegicus | |||
5. | ALA1761321 | 31 | Drug uptake | = | 0.7 | uM | ALA2396032 | uM | Rattus norvegicus | |||
6. | ALA1761313 | 22 | Drug uptake | = | 0.7 | uM | ALA2396032 | uM | Rattus norvegicus | |||
7. | ALA2391969 | 5 | Drug uptake | = | 3.4 | uM | ALA2396032 | uM | Rattus norvegicus | |||
8. | ALA373257 | 11 | Drug uptake | = | 0.2 | uM | ALA2396032 | uM | Rattus norvegicus | |||
9. | ALA478507 | 5a, JLK-1486 | Drug uptake | = | 0.037 | % | ALA3058769 | % | Rattus norvegicus | |||
10. | PF-04859989 | 7, PF-04859989 | Drug uptake | = | 4060 | nM | ALA2050759 | nM | Rattus norvegicus | |||
11. | ALA1683351 | 3 | Drug uptake | = | 85 | nM | ALA2044728 | nM | Rattus norvegicus | |||
12. | ALA2042692 | 10h | Drug uptake | = | 14 | nM | ALA2044728 | nM | Rattus norvegicus | |||
13. | ALA2042691 | 10g | Drug uptake | = | 70 | nM | ALA2044728 | nM | Rattus norvegicus | |||
14. | ALA2042690 | 10f | Drug uptake | = | 16 | nM | ALA2044728 | nM | Rattus norvegicus | |||
15. | ALA2023623 | 32 | Drug uptake | < | 1 | ng/ml | ALA2025503 | ng/ml | Rattus norvegicus | |||
16. | ALA2023457 | 14 | Drug uptake | < | 1 | ng/ml | ALA2025503 | ng/ml | Rattus norvegicus | |||
17. | ALA2022867 | 1 | Drug uptake | = | 72 | ng/ml | ALA2025336 | ng/ml | Rattus norvegicus | |||
18. | LBP-1 | 11, LBP-1 | Cmax | = | 6.4 | ng/ml | ALA2019587 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | Rattus norvegicus | ||
19. | ALA3407922 | 75 | Tmax | = | 0.5 | hr | ALA3413334 | hr | Rattus norvegicus | |||
20. | ALA3407922 | 75 | Cmax/dose | = | 0.011 | uM.kg/mg | ALA3413333 | uM.kg/mg | Rattus norvegicus |