# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA595 | Pioglitazone | Activity | 0 | ALA4433827 | Active | Rattus norvegicus | |||||
2. | L-165041 | L-165041 | Activity | 0 | ALA4433827 | Not Active | Rattus norvegicus | |||||
3. | WY-14643 (Pirinixic Acid) | 1d | Activity | 0 | ALA4433827 | Active | Rattus norvegicus | |||||
4. | ALA4449760 | 12a | Activity | 0 | ALA4433822 | Active | Rattus norvegicus | |||||
5. | ALA3407922 | 75 | t1/2 | = | 1.9 | hr | ALA3413338 | hr | Rattus norvegicus | |||
6. | ALA3407922 | 75 | Tmax | = | 0.5 | hr | ALA3413337 | hr | Rattus norvegicus | |||
7. | ALA3407922 | 75 | Cmax/dose | = | 0.03 | uM.kg/mg | ALA3413336 | uM.kg/mg | Rattus norvegicus | |||
8. | ALA3407922 | 75 | AUC/dose | = | 0.056 | uM.hr.Kg/mg | ALA3413335 | uM.hr.Kg/mg | Rattus norvegicus | |||
9. | ALA3357579 | [18F]3 | Drug uptake | 0 | ALA3386477 | Active | Rattus norvegicus | |||||
10. | ALA3357579 | [18F]3 | Drug uptake | 0 | ALA3386471 | Active | Rattus norvegicus | |||||
11. | ALA3357579 | [18F]3 | Drug uptake | 0 | ALA3386465 | Active | Rattus norvegicus | |||||
12. | ALA3354981 | [18F]1 | SUV | = | 0.2 | ALA3371791 | Rattus norvegicus | |||||
13. | ALA3354981 | [18F]1 | SUV | = | 0.5 | ALA3380944 | Rattus norvegicus | |||||
14. | ALA3354981 | [18F]1 | SUV | = | 0.19 | ALA3380940 | Rattus norvegicus | |||||
15. | ALA3354981 | [18F]1 | SUV | = | 0.51 | ALA3380936 | Rattus norvegicus | |||||
16. | ALA3354981 | [18F]1 | SUV | = | 1.7 | ALA3380932 | Rattus norvegicus | |||||
17. | ALA3597323 | (-)-[(18)F]18a | Drug uptake | = | 0.777 | % ID/g | ALA3598421 | % ID/g | Rattus norvegicus | |||
18. | ALA3589002 | 5 | Drug metabolism | 0 | ALA3592362 | metabolite_detected | Rattus norvegicus | |||||
19. | ALA3589001 | 4 | Stability | 0 | ALA3592360 | Unstable | % | Rattus norvegicus | ||||
20. | ALA3582401 | [11C]SB-216763 | Drug uptake | 0 | ALA3584788 | Active | Rattus norvegicus |