# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA2419157 | 14 | Activity | 0 | ALA4408268 | Not Active | Rattus norvegicus | |||||
2. | ALA2419157 | 14 | Activity | 0 | ALA4408269 | Active | Rattus norvegicus | |||||
3. | ALA4448829 | 42; SGE-301 | Activity | 0 | ALA4408269 | Active | Rattus norvegicus | |||||
4. | Alicapistat | 22; A-1212805, ABT-957 | INH | 0 | ALA4389025 | Active | % | Rattus norvegicus | ||||
5. | Alicapistat | 22; A-1212805, ABT-957 | IC50 | = | 385 | nM | ALA4389024 | 6.42 | nM | Rattus norvegicus | ||
6. | ALA4764801 | C01 | INH | 0 | ALA4703321 | Not Active | % | Rattus norvegicus | ||||
7. | ALA3357579 | [18F]3 | Drug uptake | 0 | ALA3386475 | Active | Rattus norvegicus | |||||
8. | ALA3357579 | [18F]3 | Drug uptake | 0 | ALA3386469 | Active | Rattus norvegicus | |||||
9. | ALA3357579 | [18F]3 | Drug uptake | 0 | ALA3385823 | Active | Rattus norvegicus | |||||
10. | ALA2441068 | 4 | Activity | 0 | ALA3389745 | Active | Rattus norvegicus | |||||
11. | ALA2441068 | 4 | Activity | 0 | ALA3389744 | Active | Rattus norvegicus | |||||
12. | ALA2441068 | 4 | Activity | 0 | ALA3389743 | Active | Rattus norvegicus | |||||
13. | ALA2441068 | 4 | Activity | 0 | ALA3389742 | Active | Rattus norvegicus | |||||
14. | ALA2441068 | 4 | Activity | 0 | ALA3389206 | Active | Rattus norvegicus | |||||
15. | ALA2441068 | 4 | Activity | 0 | ALA3389205 | Active | Rattus norvegicus | |||||
16. | ALA3358006 | 16 | Activity | 0 | ALA3383398 | Non-toxic | Rattus norvegicus | |||||
17. | ALA3358006 | 16 | Activity | 0 | ALA3383397 | Non-toxic | Rattus norvegicus | |||||
18. | ALA3358010 | 20 | Activity | 0 | ALA3383396 | Non-toxic | Rattus norvegicus | |||||
19. | ALA3358006 | 16 | Activity | 0 | ALA3383396 | Non-toxic | Rattus norvegicus | |||||
20. | ALA3358001 | 11 | Activity | 0 | ALA3383396 | Non-toxic | Rattus norvegicus |