# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | propranolol | 16 | INH | 0 | ALA3767679 | Not Active | % | Rattus norvegicus | ||||
2. | Phentolamine | Phentolamine | INH | 0 | ALA3767679 | Not Active | % | Rattus norvegicus | ||||
3. | ALA517712 | atropine | INH | 0 | ALA3767679 | Not Active | % | Rattus norvegicus | ||||
4. | Tetrodotoxin | TETRODOTOXIN | INH | 0 | ALA3767680 | Not Active | % | Rattus norvegicus | ||||
5. | ALA3335592 | 111 | Activity | 0 | ALA3378932 | Non-toxic | Rattus norvegicus | |||||
6. | ALA2297684 | 2 | Activity | 0 | ALA3378932 | Non-toxic | Rattus norvegicus | |||||
7. | Apixaban | apixaban | Papp | = | 51 | nm/s | ALA3538288 | nm/s | Rattus norvegicus | |||
8. | ALA3527012 | [14C]CS-1036 | Drug uptake | = | 33.9 | % | ALA3532512 | % | Rattus norvegicus | |||
9. | ALA3527012 | [14C]CS-1036 | Drug uptake | = | 67.7 | % | ALA3532511 | % | Rattus norvegicus | |||
10. | Neurotensin Fragment 8-13 acetate salt | NT(8-13) | EC50 | = | 3.9 | nM | ALA4737193 | 8.41 | nM | Rattus norvegicus | ||
11. | Neurotensin Fragment 8-13 acetate salt | NT(8-13) | Activity | 0 | ALA4737193 | Dose-dependent effect | Rattus norvegicus | |||||
12. | ALA4788991 | 4 | Activity | 0 | ALA4737192 | Non-Toxic | Rattus norvegicus | |||||
13. | ALA783 | 13 | Papp | = | 0.9 | 10'-4 cm/s | ALA3070491 | 10'-4 cm/s | Rattus norvegicus | |||
14. | ALA783 | 13 | Papp | = | 4.4 | 10'-4 cm/s | ALA3070485 | 10'-4 cm/s | Rattus norvegicus | |||
15. | ALA783 | 13 | Papp | = | 5.1 | 10'-4 cm/s | ALA3071418 | 10'-4 cm/s | Rattus norvegicus | |||
16. | ALA783 | 13 | Papp | = | 2 | 10'-4 cm/s | ALA3071412 | 10'-4 cm/s | Rattus norvegicus | |||
17. | ent-Nateglinide | 22 | Papp | = | 1 | 10'-4 cm/s | ALA3070491 | 10'-4 cm/s | Rattus norvegicus | |||
18. | ent-Nateglinide | 22 | Papp | = | 3.8 | 10'-4 cm/s | ALA3070485 | 10'-4 cm/s | Rattus norvegicus | |||
19. | ent-Nateglinide | 22 | Papp | = | 2.7 | 10'-4 cm/s | ALA3071418 | 10'-4 cm/s | Rattus norvegicus | |||
20. | ent-Nateglinide | 22 | Papp | = | 1.3 | 10'-4 cm/s | ALA3071412 | 10'-4 cm/s | Rattus norvegicus |