# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA2392844 | [18F]18 | SUV | = | 6.5 | % | ALA2393853 | % | Rattus norvegicus | |||
2. | ALA2391546 | 123I-CMICE-013 | Drug uptake | = | 0.846 | % ID/g | ALA2394685 | % ID/g | Rattus norvegicus | |||
3. | ALA2391546 | 123I-CMICE-013 | Drug uptake | = | 0.122 | % ID/g | ALA2394523 | % ID/g | Rattus norvegicus | |||
4. | ALA2385105 | 20 | t1/2 | > | 12 | hr | ALA2388851 | hr | Rattus norvegicus | |||
5. | ALA2387397 | 45 | t1/2 | > | 12 | hr | ALA2388851 | hr | Rattus norvegicus | |||
6. | ALA2387399 | 47 | t1/2 | > | 12 | hr | ALA2388851 | hr | Rattus norvegicus | |||
7. | ALA2387419 | 44 | t1/2 | = | 8 | hr | ALA2388851 | hr | Rattus norvegicus | |||
8. | ALA2387402 | 50 | t1/2 | 0 | ALA2388851 | Not Determined | Rattus norvegicus | |||||
9. | (3R,5R)-3-butyl-3-ethyl-7,8-dimethoxy-5-phenyl-4,5-dihydro-2H-benzo[f][1,4]thiazepine 1,1-dioxide | 2 | Stability | 0 | ALA2388858 | Unstable | % | Rattus norvegicus | ||||
10. | Linerixibat | 56, GSK2330672 | t1/2 | > | 12 | hr | ALA2388851 | hr | Rattus norvegicus | |||
11. | ALA2322005 | 25 | Peff | = | 11.28 | 10'-5cm/s | ALA2328467 | 10'-5cm/s | Rattus norvegicus | |||
12. | ALA2314493 | DTH | t1/2 | = | 168 | min | ALA2318416 | hr | Rattus norvegicus | |||
13. | ALA105592 | 2 | Stability | > | 80 | % | ALA2045897 | % | Rattus norvegicus | |||
14. | ALA105592 | 2 | Stability | > | 80 | % | ALA2045896 | % | Rattus norvegicus | |||
15. | ALA2036383 | [11C]4, [11C]2',3'-dehydropravastatin | Drug uptake | 0 | ALA2040237 | Not Active | Rattus norvegicus | |||||
16. | ALA2036383 | [11C]4, [11C]2',3'-dehydropravastatin | Drug uptake | = | 67.9 | % | ALA2040240 | % | Rattus norvegicus | |||
17. | ALA2017835 | 10e | Fu | = | 0.65 | nM | ALA2019304 | nM | Rattus norvegicus | |||
18. | ALA2017835 | 10e | Fu | = | 0.98 | nM | ALA2019303 | nM | Rattus norvegicus | |||
19. | ALA2017835 | 10e | Fu | = | 1.07 | nM | ALA2019633 | nM | Rattus norvegicus | |||
20. | Verapamil | 24 | Activity | 0 | ALA3539774 | Toxic | Rattus norvegicus |