| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA3088054 | 13, LY545694 | Cp | = | 1020 | ng/ml | ALA3089687 | ng/ml | Rattus norvegicus | |||
| 2. |  ALA3087669 | 3h | Drug metabolism | < | 5 | % | ALA3089241 | % | Rattus norvegicus | |||
| 3. | ALA3087669 | 3h | Tmax | = | 0.5 | hr | ALA3089128 | hr | Rattus norvegicus | |||
| 4. | ALA3087669 | 3h | beta t1/2 | = | 1.2 | hr | ALA3089136 | hr | Rattus norvegicus | |||
| 5. |  ALA3086991 | 1, VMY-2-95 | Fu | = | 8.4 | % | ALA3088757 | Rattus norvegicus | ||||
| 6. |  Sazetidine A dihydrochloride | 4 | Fu | = | 75.1 | % | ALA3088757 | Rattus norvegicus | ||||
| 7. |  ALA1076903 | 9a table 2 | Fu | = | 70.9 | % | ALA3088757 | Rattus norvegicus | ||||
| 8. |  propranolol | 16 | Fu | = | 9.61 | % | ALA3088757 | Rattus norvegicus | ||||
| 9. | ALA3087669 | 3h | beta t1/2 | = | 7.8 | hr | ALA3089126 | hr | Rattus norvegicus | |||
| 10. | ALA3087669 | 3h | Cmax | = | 749 | ng/ml | ALA3089130 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | Rattus norvegicus | ||
| 11. | ALA3087669 | 3h | AUC | = | 1100 | ng.hr/ml | ALA3089214 | ng.hr.mL-1 | Rattus norvegicus | |||
| 12. | ALA3087669 | 3h | AUC | = | 3150 | ng.hr/ml | ALA3089132 | ng.hr.mL-1 | Rattus norvegicus | |||
| 13. |  ALA3087342 | 25 | Drug uptake | 0 | ALA3088679 | Active | Rattus norvegicus | |||||
| 14. |  ALA3086726 | 70 | Cp(f) | = | 290 | nM | ALA3088658 | nM | Rattus norvegicus | |||
| 15. |  LY-411575 | LY-411575 | Cp(f) | = | 1.2 | nM | ALA3088658 | nM | Rattus norvegicus | |||
| 16. | LY-411575 | LY-411575 | Cp(f) | = | 0.4 | nM | ALA3088774 | nM | Rattus norvegicus | |||
| 17. | ALA3087342 | 25 | Cp(f) | = | 0.57 | nM | ALA3088411 | nM | Rattus norvegicus | |||
| 18. |  ALA3085833 | 17r | Cp | = | 0.68 | uM | ALA3089801 | uM | Rattus norvegicus | |||
| 19. | ALA3085833 | 17r | Cp | = | 5.16 | uM | ALA3089800 | uM | Rattus norvegicus | |||
| 20. |  Kisspeptin-13 (4-13) (human) (KiSS-1 (112-121)) | 10-mer, metastin-10 | Cp | = | 4.07 | nM | ALA3088602 | nM | Rattus norvegicus |
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