# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA2402081 | 37 | INH | = | 7 | % | ALA2406542 | % | Homo sapiens | |||
2. | ALA2348862 | 10b, CC214-2 | Activity | = | 95 | % | ALA2350880 | % | Homo sapiens | |||
3. | ALA2333445 | 1 | Activity | = | 95 | % | ALA2349771 | % | Homo sapiens | |||
4. | ALA2348862 | 10b, CC214-2 | Activity | = | 101 | % | ALA2350167 | % | Homo sapiens | |||
5. | ALA2348865 | 9a, CC214-1 | Activity | = | 93 | % | ALA2350880 | % | Homo sapiens | |||
6. | XL388 | 28, XL388 | IC50 | > | 10000 | nM | ALA2343437 | nM | Homo sapiens | |||
7. | ALA2012574 | 42, LDN-211898 | INH | = | 92 | % | ALA2015471 | % | Homo sapiens | |||
8. | Borussertib | EUB0000645a | % Inhibition | 15 | % | ALA4888207 | Not Active | % | Homo sapiens | |||
9. | BAY-091 | EUB0001564 | % inhibition | 11.07 | % | ALA4887990 | Not Active | % | Homo sapiens | |||
10. | BI 605906 | BI605906 | % Ctrl | 106 | % | ALA4887531 | Not Active | % | Homo sapiens | |||
11. | ALA2180408 | Figure 27, R1C1 | % inhibition | 5 | % | ALA4886311 | Not Active | % | Homo sapiens | |||
12. | ALA4475494 | 19 | % Inhibition | -6.5 | % | ALA4886050 | Not Active | % | Homo sapiens | |||
13. | ALA4097778 | 16h | pIC50 | 6 | ALA4885383 | nM | Homo sapiens | |||||
14. | ALA4549667 | EUB0000720 | pIC50 | 6 | ALA4885096 | nM | Homo sapiens | |||||
15. | ALA4088216 | 14 | pIC50 | 6 | ALA4884805 | nM | Homo sapiens | |||||
16. | ALA4580220 | EUB0000311 | % residual kinase activity | 97 | % | ALA4884423 | Not Active | % | Homo sapiens | |||
17. | Skepinone-L | 2, Skepinone-L | % Residual activity with Skepinone-L | 88 | % | ALA4884040 | Not Active | % | Homo sapiens | |||
18. | MLI-2 | 1; MLi-2 | % Inhibition | -0.099 | % | ALA4882851 | Not Active | % | Homo sapiens | |||
19. | ALA3417525 | 69, BI665915 | % Ctrl | 100.5 | % | ALA4882080 | Not Active | % | Homo sapiens | |||
20. | BAY 293 | EUB0000320 | % residual kinase activity | 84 | % | ALA4881462 | Not Active | % | Homo sapiens |