# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4083322 | 4c | Drug metabolism | 0 | ALA4013446 | Metabolite_Detected | Homo sapiens | |||||
2. | BI 2536 | 1 | Kd apparent | > | 30000 | nM | ALA3991672 | Inactive | nM | Homo sapiens | ||
3. | PF-3758309 | 1, PF-3758309 | Kd apparent | > | 30000 | nM | ALA3991672 | Inactive | nM | Homo sapiens | ||
4. | AMG-900 | SID137275938 | Kd apparent | > | 30000 | nM | ALA3991672 | Inactive | nM | Homo sapiens | ||
5. | CYC116 | 13, CYC-116 | Kd apparent | > | 30000 | nM | ALA3991672 | Inactive | nM | Homo sapiens | ||
6. | Vandetanib | 22 | Kd apparent | > | 30000 | nM | ALA3991672 | Inactive | nM | Homo sapiens | ||
7. | GSK2636771 | SID174006492 | Kd apparent | > | 30000 | nM | ALA3991672 | Inactive | nM | Homo sapiens | ||
8. | Tozasertib | VX-680 | Kd apparent | > | 30000 | nM | ALA3991672 | Inactive | nM | Homo sapiens | ||
9. | Tucatinib (Irbinitinib, ONT-380) | TUCATINIB | Kd apparent | > | 30000 | nM | ALA3991672 | Inactive | nM | Homo sapiens | ||
10. | ALA1614701 | AZD-6244 | Kd apparent | > | 30000 | nM | ALA3991672 | Inactive | nM | Homo sapiens | ||
11. | Dabrafenib | 7, GSK2118436 | Kd apparent | > | 30000 | nM | ALA3991672 | Inactive | nM | Homo sapiens | ||
12. | RGB-286638 | RGB-286638 | Kd apparent | > | 30000 | nM | ALA3991672 | Inactive | nM | Homo sapiens | ||
13. | LY2584702 | LY-2584702 | Kd apparent | > | 30000 | nM | ALA3991672 | Inactive | nM | Homo sapiens | ||
14. | P276-00 | P-276-00 | Kd apparent | > | 30000 | nM | ALA3991672 | Inactive | nM | Homo sapiens | ||
15. | AZD7762 | AZD-7762 | Kd apparent | > | 30000 | nM | ALA3991672 | Inactive | nM | Homo sapiens | ||
16. | Barasertib (AZD1152-HQPA) | 34 | Kd apparent | > | 30000 | nM | ALA3991672 | Inactive | nM | Homo sapiens | ||
17. | Masitinib (AB1010) | AB-1010 | Kd apparent | > | 30000 | nM | ALA3991672 | Inactive | nM | Homo sapiens | ||
18. | PHA-793887 | 31 | Kd apparent | > | 30000 | nM | ALA3991672 | Inactive | nM | Homo sapiens | ||
19. | Linifanib (ABT-869) | 17p, ABT-869 | Kd apparent | = | 6 | nM | ALA3991672 | 8.22 | Uncertain | nM | Homo sapiens | |
20. | ALA3184679 | AZD-4547 | Kd apparent | > | 30000 | nM | ALA3991672 | Inactive | nM | Homo sapiens |