# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA3261993 | [11C]1 | Kd | = | 1.25 | nM | ALA5235640 | 8.90 | nM | Rattus norvegicus | ||
2. | ALA5272386 | [11C]KIT-6; [11C]T-773 | Kd | = | 4.7 | nmol/L | ALA5235634 | 8.33 | nM | Rattus norvegicus | ||
3. | ALA5272386 | [11C]KIT-6; [11C]T-773 | Kd | = | 12.2 | nmol/L | ALA5235633 | 7.91 | nM | Rattus norvegicus | ||
4. | ALA3092563 | 19, [18F]-19 | IC50 | = | 14 | nM | ALA5227559 | 7.85 | nM | Rattus norvegicus | ||
5. | ALA5266641 | [11C]Lu AE92686 | IC50 | = | 0.39 | nM | ALA5227559 | 9.41 | nM | Rattus norvegicus | ||
6. | Papaverine | Papaverine | IC50 | = | 36 | nM | ALA4339834 | 7.44 | nM | Rattus norvegicus | ||
7. | Papaverine | Papaverine | IC50 | = | 36 | nM | ALA4231524 | 7.44 | nM | Rattus norvegicus | ||
8. | ALA4785227 | 40 | IC50 | = | 8318 | nM | ALA4672634 | 5.08 | nM | Rattus norvegicus | ||
9. | ALA4797527 | 39 | IC50 | = | 5623 | nM | ALA4672634 | 5.25 | nM | Rattus norvegicus | ||
10. | ALA4758766 | 38 | IC50 | = | 7586 | nM | ALA4672634 | 5.12 | nM | Rattus norvegicus | ||
11. | ALA4776046 | 37 | IC50 | = | 661 | nM | ALA4672634 | 6.18 | nM | Rattus norvegicus | ||
12. | ALA4780124 | 36 | IC50 | = | 550 | nM | ALA4672634 | 6.26 | nM | Rattus norvegicus | ||
13. | ALA4757440 | 35 | IC50 | = | 100 | nM | ALA4672634 | 7.00 | nM | Rattus norvegicus | ||
14. | ALA4745282 | 34 | IC50 | > | 10000 | nM | ALA4672634 | nM | Rattus norvegicus | |||
15. | ALA4764226 | 33 | IC50 | = | 1096 | nM | ALA4672634 | 5.96 | nM | Rattus norvegicus | ||
16. | ALA4751598 | 32 | IC50 | = | 724 | nM | ALA4672634 | 6.14 | nM | Rattus norvegicus | ||
17. | ALA4755779 | 31 | IC50 | = | 912 | nM | ALA4672634 | 6.04 | nM | Rattus norvegicus | ||
18. | ALA4793092 | 30 | IC50 | = | 2692 | nM | ALA4672634 | 5.57 | nM | Rattus norvegicus | ||
19. | ALA4761452 | 29 | IC50 | = | 759 | nM | ALA4672634 | 6.12 | nM | Rattus norvegicus | ||
20. | ALA4746828 | 28 | IC50 | = | 1148 | nM | ALA4672634 | 5.94 | nM | Rattus norvegicus |