# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA2402081 | 37 | INH | = | 6 | % | ALA2405115 | % | Homo sapiens | |||
2. | ALA2348862 | 10b, CC214-2 | Activity | = | 103 | % | ALA2352891 | % | Homo sapiens | |||
3. | ALA2333445 | 1 | Activity | = | 97 | % | ALA2352181 | % | Homo sapiens | |||
4. | ALA2348862 | 10b, CC214-2 | Activity | = | 94 | % | ALA2351969 | % | Homo sapiens | |||
5. | ALA2348865 | 9a, CC214-1 | Activity | = | 102 | % | ALA2352891 | % | Homo sapiens | |||
6. | Borussertib | EUB0000645a | % Inhibition | 2 | % | ALA4888183 | Not Active | % | Homo sapiens | |||
7. | BAY-091 | EUB0001564 | % inhibition | 0.16 | % | ALA4887884 | Not Active | % | Homo sapiens | |||
8. | BI 605906 | BI605906 | % Ctrl | 93 | % | ALA4887440 | Not Active | % | Homo sapiens | |||
9. | ALA2180408 | Figure 27, R1C1 | % inhibition | 3 | % | ALA4886241 | Not Active | % | Homo sapiens | |||
10. | ALA4475494 | 19 | % Inhibition | 3.5 | % | ALA4885983 | Not Active | % | Homo sapiens | |||
11. | ALA4097778 | 16h | pIC50 | 6 | ALA4885303 | nM | Homo sapiens | |||||
12. | ALA4549667 | EUB0000720 | pIC50 | 6 | ALA4885012 | nM | Homo sapiens | |||||
13. | ALA4088216 | 14 | pIC50 | 6 | ALA4884721 | nM | Homo sapiens | |||||
14. | ALA4580220 | EUB0000311 | % residual kinase activity | 96 | % | ALA4884325 | Not Active | % | Homo sapiens | |||
15. | Skepinone-L | 2, Skepinone-L | % Residual activity with Skepinone-L | 82 | % | ALA4883939 | Not Active | % | Homo sapiens | |||
16. | MLI-2 | 1; MLi-2 | % Inhibition | 6.633 | % | ALA4882751 | Not Active | % | Homo sapiens | |||
17. | ALA3417525 | 69, BI665915 | % Ctrl | 101.5 | % | ALA4881980 | Not Active | % | Homo sapiens | |||
18. | BAY-885 | BAY-885; 41 | % residual kinase activity | 111 | % | ALA4881066 | Not Active | % | Homo sapiens | |||
19. | 2,6-Dimethyl-4-(3-methyl-1H-indazol-5-yl)-1,4-dihydropyridine-3,5-dicarbonitrile(BAY-474) | EUB0000293 | % inhibition | -2 | % | ALA4880640 | Not Active | % | Homo sapiens | |||
20. | ALA3298678 | 38 | INH | = | 4.5 | % | ALA3366830 | % | Homo sapiens |