# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5284303 | R-26j; RK-0133114 | IC50 | = | 53 | nM | ALA5251533 | 7.28 | nM | Homo sapiens | ||
2. | ALA5266889 | 9; DS79932728 | IC50 | = | 75.7 | nM | ALA5251533 | 7.12 | nM | Homo sapiens | ||
3. | A 366 | 12, A-366 | IC50 | = | 38 | nM | ALA5251533 | 7.42 | nM | Homo sapiens | ||
4. | UNC 0642 | 7, UNC0642 | IC50 | < | 2.5 | nM | ALA5251533 | nM | Homo sapiens | |||
5. | UNC0638 | 5, UNC0638 | IC50 | = | 19 | nM | ALA5251533 | 7.72 | nM | Homo sapiens | ||
6. | SGC 0946 | 24, SGC0946 | IC50 | > | 100 | uM | ALA5214639 | nM | Homo sapiens | |||
7. | (R)-PFI 2 hydrochloride | EUB0000196bCl | EC50 | > | 10 | uM | ALA5214703 | nM | Homo sapiens | |||
8. | OICR-9429 | 16d; OICR-9429 | % activity remaining | > | 90 | % | ALA5213718 | % | Homo sapiens | |||
9. | A 366 | 12, A-366 | IC50 | = | 38 | nM | ALA5210607 | 7.42 | nM | Homo sapiens | ||
10. | UNC 0642 | 7, UNC0642 | IC50 | < | 2.5 | nM | ALA5210589 | nM | Homo sapiens | |||
11. | A 366 | 12, A-366 | EC50 | < | 3000 | nM | ALA5210103 | nM | Homo sapiens | |||
12. | UNC 0642 | 7, UNC0642 | IC50 | = | 106 | nM | ALA5210096 | 6.97 | nM | Homo sapiens | ||
13. | ALA5191361 | D7 | INH | 0 | ALA5144729 | Active | % | Homo sapiens | ||||
14. | UNC 0642 | 7, UNC0642 | IC50 | = | 2.8 | nM | ALA5144717 | 8.55 | nM | Homo sapiens | ||
15. | ALA5206158 | D8 | IC50 | = | 190 | nM | ALA5144717 | 6.72 | nM | Homo sapiens | ||
16. | ALA5191361 | D7 | IC50 | = | 1.3 | nM | ALA5144717 | 8.89 | nM | Homo sapiens | ||
17. | ALA5201140 | D6 | IC50 | = | 9.2 | nM | ALA5144717 | 8.04 | nM | Homo sapiens | ||
18. | ALA5171820 | D5 | IC50 | = | 1.6 | nM | ALA5144717 | 8.80 | nM | Homo sapiens | ||
19. | ALA5204152 | D4 | IC50 | = | 11 | nM | ALA5144717 | 7.96 | nM | Homo sapiens | ||
20. | ALA5171881 | D3 | IC50 | = | 97 | nM | ALA5144717 | 7.01 | nM | Homo sapiens |