| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  CHMFL-FLT3-122 | 18; CHMFL-FLT3-122 | Activity | = | 0.05 | % | ALA3749070 | % | Homo sapiens | |||
| 2. |  ALA5284848 | 14d | Activity | 0 | ALA5250209 | Active | Homo sapiens | |||||
| 3. |  ALA5282275 | 12; TX1-121-1 | IC50 | = | 49 | nM | ALA5243474 | 7.31 | nM | Homo sapiens | ||
| 4. |  ALA5285282 | 11; TX1-85-1 | IC50 | = | 23 | nM | ALA5243474 | 7.64 | nM | Homo sapiens | ||
| 5. |  ALA3969370 | 19; FMF-01-086-2 | Activity | = | 81 | % | ALA4185796 | % | Homo sapiens | |||
| 6. |  ALA4206831 | 2; FMF-03-145-1 | Activity | = | 85 | % | ALA4185796 | % | Homo sapiens | |||
| 7. |  mavelertinib | MAVELERTINIB | Ratio | = | 68000 | /M/s | ALA4178442 | /M/s | Homo sapiens | |||
| 8. |  PF-06459988 | 1; PF-06459988 | IC50 | = | 21 | nM | ALA4178362 | 7.68 | nM | Homo sapiens | ||
| 9. |  PF 6274484 | PF-6274484 | IC50 | = | 1 | nM | ALA4178362 | 9.00 | nM | Homo sapiens | ||
| 10. |  Erlotinib | Tarceva | IC50 | = | 10 | nM | ALA4178362 | 8.00 | nM | Homo sapiens | ||
| 11. |  CO-1686 (AVL-301) | ROCILETINIB | IC50 | = | 46 | nM | ALA4178362 | 7.34 | nM | Homo sapiens | ||
| 12. |  ALA4206501 | 23; AZD9291 | IC50 | = | 36 | nM | ALA4178362 | 7.44 | nM | Homo sapiens | ||
| 13. | mavelertinib | MAVELERTINIB | IC50 | = | 4 | nM | ALA4178362 | 8.40 | nM | Homo sapiens | ||
| 14. |  ALA4218154 | 17 | IC50 | 0 | ALA4178362 | Not Determined | Homo sapiens | |||||
| 15. |  ALA4216679 | 16 | IC50 | = | 2 | nM | ALA4178362 | 8.70 | nM | Homo sapiens | ||
| 16. |  ALA3608432 | 61 | IC50 | = | 9 | nM | ALA4178362 | 8.05 | nM | Homo sapiens | ||
| 17. |  ALA3608429 | 2 | IC50 | = | 2 | nM | ALA4178362 | 8.70 | nM | Homo sapiens | ||
| 18. |  ALA4174988 | 15i | Activity | = | 95 | % | ALA4157017 | % | Homo sapiens | |||
| 19. | ALA4174988 | 15i | Activity | = | 79 | % | ALA4156997 | % | Homo sapiens | |||
| 20. |  Ibrutinib (PCI-32765) | SID124898784 | GI50 | = | 0.004 | uM | ALA4130930 | nM | Homo sapiens |
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