# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | N-(4-{3-[2-(methylcarbamoyl)ethyl]-5-[4'-(trifluoromethyl)-[1,1'-biphenyl]-4-yl]-1H-pyrazol-1-yl}phenyl)prop-2-ynamide | 1; Tr-87 | Activity | 0 | ALA4415378 | Active | Homo sapiens | |||||
2. | ALA3359147 | 4a | Ki | = | 4.3 | uM | ALA3374599 | 5.37 | nM | Homo sapiens | ||
3. | LW 6 | 23 | Ki | = | 1.9 | uM | ALA3374599 | 5.72 | nM | Homo sapiens | ||
4. | ALA3359147 | 4a | INH | 0 | ALA3374598 | Active | % | Homo sapiens | ||||
5. | LW 6 | 23 | INH | 0 | ALA3374598 | Active | % | Homo sapiens | ||||
6. | ALA3359147 | 4a | INH | 0 | ALA3374597 | Active | % | Homo sapiens | ||||
7. | LW 6 | 23 | INH | 0 | ALA3374597 | Active | % | Homo sapiens | ||||
8. | ALA3359148 | 4b | Activity | 0 | ALA3374594 | Not Active | Homo sapiens | |||||
9. | ALA3359147 | 4a | Activity | 0 | ALA3374594 | Active | Homo sapiens | |||||
10. | ALA3359146 | 4j | Activity | 0 | ALA3374594 | Not Active | Homo sapiens | |||||
11. | ALA3359145 | 4i | Activity | 0 | ALA3374594 | Active | Homo sapiens | |||||
12. | ALA3359142 | 4f | Activity | 0 | ALA3374594 | Not Active | Homo sapiens | |||||
13. | ALA3359141 | 4e | Activity | 0 | ALA3374594 | Not Active | Homo sapiens | |||||
14. | ALA3359141 | 4e | Activity | 0 | ALA3374591 | Active | Homo sapiens | |||||
15. | ALA3359148 | 4b | IC50 | > | 20 | uM | ALA3374593 | nM | Homo sapiens | |||
16. | ALA3359147 | 4a | IC50 | = | 5.5 | uM | ALA3374593 | 5.26 | nM | Homo sapiens | ||
17. | ALA3359146 | 4j | IC50 | > | 20 | uM | ALA3374593 | nM | Homo sapiens | |||
18. | ALA3359145 | 4i | IC50 | = | 10.2 | uM | ALA3374593 | 4.99 | nM | Homo sapiens | ||
19. | ALA3359144 | 4h | IC50 | > | 20 | uM | ALA3374593 | nM | Homo sapiens | |||
20. | ALA3359143 | 4g | IC50 | > | 20 | uM | ALA3374593 | nM | Homo sapiens |