# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA3480577 | DDD01251909 | Mean fold stimulation | 1.025 | ALA4883546 | Homo sapiens | ||||||
2. | ALA3422018 | 39 | INH | = | 24 | % | ALA3425014 | % | Homo sapiens | |||
3. | ALA3422010 | 31 | INH | = | 18 | % | ALA3425014 | % | Homo sapiens | |||
4. | ALA3422009 | 3 | INH | = | -14 | % | ALA3425014 | % | Homo sapiens | |||
5. | ALA3422516 | 17 | EC50 | = | 222 | nM | ALA3423987 | 6.65 | nM | Homo sapiens | ||
6. | ALA3422408 | 3 | EC50 | > | 5 | uM | ALA3423987 | nM | Homo sapiens | |||
7. | ALA3422407 | 2 | EC50 | > | 5 | uM | ALA3423987 | nM | Homo sapiens | |||
8. | ALA3361415 | 17g | Ki | = | 2348 | nM | ALA3387184 | 5.63 | nM | Homo sapiens | ||
9. | ALA3361414 | 17f | Ki | = | 1966 | nM | ALA3387184 | 5.71 | nM | Homo sapiens | ||
10. | ALA3361413 | 17e | Ki | = | 1623 | nM | ALA3387184 | 5.79 | nM | Homo sapiens | ||
11. | ALA3361412 | 17d | Ki | = | 2454 | nM | ALA3387184 | 5.61 | nM | Homo sapiens | ||
12. | ALA3352907 | 17c | Ki | = | 2692 | nM | ALA3387184 | 5.57 | nM | Homo sapiens | ||
13. | ALA3361433 | 53a | Activity | 0 | ALA3387755 | Dose-dependent effect | Homo sapiens | |||||
14. | 4-anilino-1-benzyl-N-[2-(diaminomethylideneamino)ethyl]piperidine-4-carboxamide | 46 | Activity | 0 | ALA3387755 | Dose-dependent effect | Homo sapiens | |||||
15. | ALA3360829 | RF9 | Emax | = | 79 | % | ALA3388430 | % | Homo sapiens | |||
16. | ALA3361433 | 53a | Emax | = | 56.2 | % | ALA3387755 | % | Homo sapiens | |||
17. | 4-anilino-1-benzyl-N-[2-(diaminomethylideneamino)ethyl]piperidine-4-carboxamide | 46 | Emax | = | 68 | % | ALA3387755 | % | Homo sapiens | |||
18. | ALA3361416 | 21 | Emax | = | 83 | % | ALA3387755 | % | Homo sapiens | |||
19. | ALA3360829 | RF9 | EC50 | = | 4700 | nM | ALA3388430 | 5.33 | nM | Homo sapiens | ||
20. | ALA3361433 | 53a | Ratio EC50 | = | 12 | ALA3387760 | Homo sapiens |