# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4873511 | 3x-SEE | Activity | = | 26 | pmol/min/mg | ALA4841950 | pmol/min/mg | Homo sapiens | |||
2. | ALA4868959 | 3x-FEE | Activity | = | 29.5 | pmol/min/mg | ALA4841950 | pmol/min/mg | Homo sapiens | |||
3. | ALA4853566 | 3w-SEE | Activity | = | 16.3 | pmol/min/mg | ALA4841950 | pmol/min/mg | Homo sapiens | |||
4. | ALA4870172 | 3w-FEE | Activity | = | 10.2 | pmol/min/mg | ALA4841950 | pmol/min/mg | Homo sapiens | |||
5. | ALA4877554 | 3v-SEE | Activity | = | 39.7 | pmol/min/mg | ALA4841950 | pmol/min/mg | Homo sapiens | |||
6. | ALA4849286 | 3v-FEE | Activity | = | 30.3 | pmol/min/mg | ALA4841950 | pmol/min/mg | Homo sapiens | |||
7. | ALA4848092 | 3l-SEE | Activity | = | 33.6 | pmol/min/mg | ALA4841950 | pmol/min/mg | Homo sapiens | |||
8. | ALA4854086 | 3l-FEE | Activity | = | 35.9 | pmol/min/mg | ALA4841950 | pmol/min/mg | Homo sapiens | |||
9. | Tenofovir alafenamide fumarate | TAF | Activity | = | 25.8 | pmol/min/mg | ALA4841950 | pmol/min/mg | Homo sapiens | |||
10. | vaborbactam | 27, RPX7009 | IC50 | = | 1000 | uM | ALA3578763 | nM | Homo sapiens | |||
11. | Carfilzomib | 2 | IC50 | > | 30 | uM | ALA3240090 | nM | Homo sapiens | |||
12. | ALA3237873 | 11a | IC50 | > | 30 | uM | ALA3240090 | nM | Homo sapiens | |||
13. | ALA3237863 | 4a | IC50 | > | 30 | uM | ALA3240090 | nM | Homo sapiens | |||
14. | Bortezomib (PS-341) | 15 | IC50 | = | 9.2 | uM | ALA3240090 | 5.04 | nM | Homo sapiens | ||
15. | ALA3955075 | BDBM193646 | IC50 | = | 4942 | nM | ALA3887623 | 5.31 | 345969 | nM | Homo sapiens | |
16. | ALA3966115 | BDBM193645 | IC50 | = | 935 | nM | ALA3887623 | 6.03 | 345968 | nM | Homo sapiens | |
17. | ALA3914838 | BDBM193523 | IC50 | = | 20600 | nM | ALA3887623 | 4.69 | 345967 | nM | Homo sapiens | |
18. | ALA3970600 | BDBM193643 | IC50 | = | 6710 | nM | ALA3887623 | 5.17 | 345966 | nM | Homo sapiens | |
19. | ALA3931940 | BDBM193642 | IC50 | = | 4740 | nM | ALA3887623 | 5.32 | 345965 | nM | Homo sapiens | |
20. | ALA3932858 | BDBM193641 | IC50 | = | 1720 | nM | ALA3887623 | 5.76 | 345964 | nM | Homo sapiens |