| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  4-[4-[3-(1H-pyrazol-4-yl)pyrazolo[1,5-a]pyrimidin-6-yl]phenyl]morpholine | 13a | IC50 | = | 39.9 | nM | ALA2390519 | 7.40 | nM | Homo sapiens | ||
| 2. |  ALA2385600 | 7d | IC50 | = | 44 | nM | ALA2390519 | 7.36 | nM | Homo sapiens | ||
| 3. |  ALA2385586 | 13h | IC50 | = | 82 | nM | ALA2390519 | 7.09 | nM | Homo sapiens | ||
| 4. |  Dorsomorphin | 1 | IC50 | = | 234.6 | nM | ALA2390519 | 6.63 | nM | Homo sapiens | ||
| 5. |  4-[6-[4-(4-methylpiperazin-1-yl)phenyl]pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | 13r | IC50 | = | 960 | nM | ALA2390519 | 6.02 | nM | Homo sapiens | ||
| 6. |  LDN-193189 | 13 | IC50 | = | 1122 | nM | ALA2390519 | 5.95 | nM | Homo sapiens | ||
| 7. |  LDN 212854 | 13m | IC50 | = | 2520 | nM | ALA2390519 | 5.60 | nM | Homo sapiens | ||
| 8. |  4-[4-(3-quinolin-4-ylpyrazolo[1,5-a]pyrimidin-6-yl)phenyl]morpholine | 13d | IC50 | = | 2680 | nM | ALA2390519 | 5.57 | nM | Homo sapiens | ||
| 9. |  ALA511563 | 52 | IC50 | = | 7260 | nM | ALA2390519 | 5.14 | nM | Homo sapiens | ||
| 10. |  DMH-1 | 3, DMH1, VU0364852 | IC50 | 0 | ALA2390519 | Not Active | Homo sapiens | |||||
| 11. |  ML 347 | 50 | IC50 | 0 | ALA2390519 | Not Active | Homo sapiens | |||||
| 12. |  XL388 | 28, XL388 | IC50 | > | 10000 | nM | ALA2343944 | nM | Homo sapiens | |||
| 13. |  Khk-IN-1 | 8 | IC50 | > | 40 | uM | ALA2019660 | nM | Homo sapiens | |||
| 14. |  MK-8722 | 6; MK-8722 | Activity | 0 | ALA4828043 | Not Active | Homo sapiens | |||||
| 15. |  ALA4094080 | 19 | INH | = | 17 | % | ALA4048662 | % | Homo sapiens | |||
| 16. |  MARK4 inhibitor 1 | 9g | INH | 0 | ALA4412652 | Not Active | % | Homo sapiens | ||||
| 17. |  ALA4462318 | 19i | Kd(free) | = | 2.279 | uM | ALA4371429 | 5.64 | nM | Homo sapiens | ||
| 18. |  ALA4443828 | 19h | Kd(free) | = | 1.257 | uM | ALA4371429 | 5.90 | nM | Homo sapiens | ||
| 19. |  ALA3950376 | 15 | EC50 | < | 500 | nM | ALA3859849 | nM | Homo sapiens | |||
| 20. |  ALA3979403 | 16; 17 | Activity | = | 132 | % | ALA3859852 | % | Homo sapiens |
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