# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4083190 | Ac-KISQLD-aldehyde | IC50 | > | 100 | uM | ALA3992262 | nM | Homo sapiens | |||
2. | ALA4101191 | Ac-ISQLD-cmk | IC50 | > | 100 | uM | ALA3992262 | nM | Homo sapiens | |||
3. | yzm18 | yzm18, Ac-Ile-Ser-Gln-Leu-Asp-vs | IC50 | = | 29.4 | uM | ALA3992262 | 4.53 | nM | Homo sapiens | ||
4. | ALA1091971 | NSC-48300 | IC50 | = | 7.5 | uM | ALA3992262 | 5.12 | nM | Homo sapiens | ||
5. | Bortezomib (PS-341) | 15 | INH | 0 | ALA3992263 | Not Active | % | Homo sapiens | ||||
6. | ALA1091971 | NSC-48300 | INH | 0 | ALA3992264 | Active | % | Homo sapiens | ||||
7. | ALA1091971 | NSC-48300 | INH | 0 | ALA3992266 | Active | % | Homo sapiens | ||||
8. | ALA2374288 | SID573565 | INH | 0 | ALA3992267 | Not Active | % | Homo sapiens | ||||
9. | ALA1091971 | NSC-48300 | INH | 0 | ALA3992268 | Not Active | % | Homo sapiens | ||||
10. | ALA4090722 | NSC74084 | INH | 0 | ALA3992269 | Not Active | % | Homo sapiens | ||||
11. | ALA4069728 | NSC49855 | INH | 0 | ALA3992269 | Not Active | % | Homo sapiens | ||||
12. | ALA1091971 | NSC-48300 | Ki | = | 4.22 | uM | ALA3992273 | 5.38 | nM | Homo sapiens | ||
13. | ALA4072434 | SPB08132 | EC50 | = | 5.9 | uM | ALA3992283 | 5.23 | nM | Homo sapiens | ||
14. | ALA4061045 | BTB00807 | EC50 | = | 9.9 | uM | ALA3992283 | 5.00 | nM | Homo sapiens | ||
15. | ALA4083855 | HTS01888 | EC50 | = | 2.2 | uM | ALA3992283 | 5.66 | nM | Homo sapiens | ||
16. | ALA3758545 | 3; NS-00432073 | EC50 | = | 4 | uM | ALA3992283 | 5.40 | nM | Homo sapiens | ||
17. | ALA4091631 | CD02506 | EC50 | = | 1.5 | uM | ALA3992283 | 5.82 | nM | Homo sapiens | ||
18. | ALA4063845 | CD06082 | EC50 | = | 3.3 | uM | ALA3992283 | 5.48 | nM | Homo sapiens | ||
19. | ALA4099366 | RJF02020 | EC50 | = | 3.9 | uM | ALA3992283 | 5.41 | nM | Homo sapiens | ||
20. | ALA570439 | yzm38 | IC50 | > | 100 | uM | ALA1042727 | nM | Homo sapiens |