# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | 4-Aminocinnoline-3-carboxamide | HTS-9026 | Kd | = | 300 | nM | ALA5252740 | 6.52 | nM | Homo sapiens | ||
2. | ALA3586447 | 11 | INH | = | 71 | % | ALA5252737 | % | Homo sapiens | |||
3. | ALA3586443 | 7 | INH | = | 94.4 | % | ALA5252737 | % | Homo sapiens | |||
4. | 4-Aminocinnoline-3-carboxamide | HTS-9026 | INH | = | 88 | % | ALA5252737 | % | Homo sapiens | |||
5. | Defactinib | DEFACTINIB | % of control | = | 1.7 | % | ALA5213441 | % | Homo sapiens | |||
6. | ALA4518706 | EUB0000702 | % of control | = | 0.4 | % | ALA5213320 | % | Homo sapiens | |||
7. | BAY-985 | 34; BAY-985 | IC50 | > | 20 | uM | ALA5213269 | nM | Homo sapiens | |||
8. | BAY-985 | 34; BAY-985 | % of control | = | 10 | % | ALA5213268 | % | Homo sapiens | |||
9. | BAY-985 | 34; BAY-985 | Kd | = | 9.6 | nM | ALA5213267 | 8.02 | nM | Homo sapiens | ||
10. | ALA4538591 | 36; BAY-440 | % of control | = | 15 | % | ALA5213294 | % | Homo sapiens | |||
11. | ALA4799297 | EUB0000589aTFA | Kd | = | 200 | nM | ALA5214798 | 6.70 | nM | Homo sapiens | ||
12. | ALA5190298 | 22 | INH | = | 96 | % | ALA5149693 | % | Homo sapiens | |||
13. | ALA3979678 | BDBM238766 | Activity | = | 0.4 | % | ALA4478503 | % | Homo sapiens | |||
14. | ALA4455923 | 48c | INH | < | 50 | % | ALA4405620 | % | Homo sapiens | |||
15. | ALA4559936 | (+/-)-6 | Activity | = | 8.5 | % | ALA4391647 | % | Homo sapiens | |||
16. | ALA4564973 | 50 | INH | = | 40 | % | ALA4390021 | % | Homo sapiens | |||
17. | ALA4555459 | 43 | INH | = | 2.3 | % | ALA4389544 | % | Homo sapiens | |||
18. | ALA4473365 | 7c | Activity | = | 14 | % | ALA4382825 | % | Homo sapiens | |||
19. | BAY-985 | 34; BAY-985 | INH | 0 | ALA4380558 | Active | % | Homo sapiens | ||||
20. | ALA4435393 | 24 | INH | 0 | ALA4380558 | Active | % | Homo sapiens |