| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  Pitolisant | BF2.649 | Ki | = | 13.4 | uM | ALA5240507 | 4.87 | nM | Homo sapiens | ||
| 2. |  ALA5265920 | LINS050021 | Ki | = | 0.91 | uM | ALA5240507 | 6.04 | nM | Homo sapiens | ||
| 3. |  ALA5278711 | LINS050020 | Ki | = | 0.27 | uM | ALA5240507 | 6.57 | nM | Homo sapiens | ||
| 4. |  ALA5287235 | LINS050019 | Ki | = | 1.7 | uM | ALA5240507 | 5.77 | nM | Homo sapiens | ||
| 5. |  ALA5270288 | LINS050018 | Ki | = | 3.3 | uM | ALA5240507 | 5.48 | nM | Homo sapiens | ||
| 6. |  ALA5276588 | LINS050016 | Ki | = | 1.9 | uM | ALA5240507 | 5.72 | nM | Homo sapiens | ||
| 7. |  ALA5270151 | LINS050015 | Ki | = | 1.1 | uM | ALA5240507 | 5.96 | nM | Homo sapiens | ||
| 8. |  ALA5282002 | LINS050014 | Ki | = | 3.7 | uM | ALA5240507 | 5.43 | nM | Homo sapiens | ||
| 9. |  ALA5283987 | LINS050011 | Ki | = | 2.2 | uM | ALA5240507 | 5.66 | nM | Homo sapiens | ||
| 10. |  ALA5289654 | LINS05009 | Ki | 0 | ALA5240507 | Not Determined | Homo sapiens | |||||
| 11. |  ALA4293814 | 14 | Ki | > | 10 | uM | ALA5240507 | nM | Homo sapiens | |||
| 12. |  ALA5289468 | LINS05007 | Ki | = | 4 | uM | ALA5240507 | 5.40 | nM | Homo sapiens | ||
| 13. |  ALA5280702 | LINS05006 | Ki | = | 2.8 | uM | ALA5240507 | 5.55 | nM | Homo sapiens | ||
| 14. |  ALA5267271 | LINS05005 | Ki | 0 | ALA5240507 | Not Determined | Homo sapiens | |||||
| 15. |  ALA5276899 | LINS05001 | Ki | 0 | ALA5240507 | Not Determined | Homo sapiens | |||||
| 16. | Pitolisant | BF2.649 | INH | = | 99.8 | % | ALA5240501 | % | Homo sapiens | |||
| 17. | ALA5265920 | LINS050021 | INH | = | 80.5 | % | ALA5240500 | % | Homo sapiens | |||
| 18. | ALA5278711 | LINS050020 | INH | = | 88.8 | % | ALA5240500 | % | Homo sapiens | |||
| 19. | ALA5289654 | LINS05009 | INH | = | 54 | % | ALA5240500 | % | Homo sapiens | |||
| 20. | ALA4293814 | 14 | INH | = | 36.8 | % | ALA5240500 | % | Homo sapiens |
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