# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4541720 | CKI-E | INH | = | 25 | % | ALA4370858 | % | Mus musculus | |||
2. | ALA4454648 | CKI-F | INH | = | 30 | % | ALA4370858 | % | Mus musculus | |||
3. | Odanacatib (MK-0822) | 24, odanacatib | INH | = | 19 | % | ALA4370858 | % | Mus musculus | |||
4. | ALA4541720 | CKI-E | INH | 0 | ALA4370860 | Active | % | Mus musculus | ||||
5. | ALA4454648 | CKI-F | INH | 0 | ALA4370860 | Active | % | Mus musculus | ||||
6. | Odanacatib (MK-0822) | 24, odanacatib | INH | 0 | ALA4370860 | Active | % | Mus musculus | ||||
7. | ALA251719 | 21 | IC50 | = | 2553 | nM | ALA923080 | 5.59 | nM | Mus musculus | ||
8. | ALA400387 | 2 | IC50 | = | 1030 | nM | ALA923080 | 5.99 | nM | Mus musculus | ||
9. | ALA249915 | 6 | IC50 | = | 1646 | nM | ALA923080 | 5.78 | nM | Mus musculus | ||
10. | ALA250119 | 7 | IC50 | = | 5835 | nM | ALA923080 | 5.23 | nM | Mus musculus | ||
11. | ALA251327 | 12 | IC50 | > | 10000 | nM | ALA923080 | nM | Mus musculus | |||
12. | ALA400750 | 15 | IC50 | > | 10000 | nM | ALA923080 | nM | Mus musculus | |||
13. | ALA250720 | 20 | IC50 | = | 1324 | nM | ALA923080 | 5.88 | nM | Mus musculus | ||
14. | ALA443319 | 24 | IC50 | = | 1464 | nM | ALA923080 | 5.83 | nM | Mus musculus | ||
15. | LHVS | LHVS | IC50 | = | 388 | nM | ALA923080 | 6.41 | nM | Mus musculus | ||
16. | L-873724 | 22 | IC50 | = | 43 | nM | ALA923080 | 7.37 | nM | Mus musculus |