# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4095790 | Table 2, R4C1 | Ratio | = | 25 | ALA4049740 | Rattus norvegicus | |||||
2. | ALA4077758 | Table 2, R5C1 | Ratio | = | 11 | ALA4049740 | Rattus norvegicus | |||||
3. | ALA4095790 | Table 2, R4C1 | Ratio | = | 25 | ALA4049752 | Rattus norvegicus | |||||
4. | ALA4077758 | Table 2, R5C1 | Ratio | = | 11 | ALA4049752 | Rattus norvegicus | |||||
5. | 5-Hydroxytryptamine | 1a | Activity | 0 | ALA2078187 | is not an inhibitor [-] | Rattus norvegicus | |||||
6. | L-Noradrenaline | NE | Activity | 0 | ALA2078189 | is not an inhibitor [-] | Rattus norvegicus | |||||
7. | guanidine | 14 | Activity | 0 | ALA2078194 | is not an inhibitor [-] | Rattus norvegicus | |||||
8. | Ceftazidime | CAZ | Activity | 0 | ALA2078208 | is not an inhibitor [-] | Rattus norvegicus | |||||
9. | Cefadroxil | 85(Cefadroxil) | Activity | 0 | ALA2078212 | is not an inhibitor [-] | Rattus norvegicus | |||||
10. | tetraethylammonium | 1 | Km | = | 63 | uM | ALA2076296 | substrate [Km=63uM] | nM | Rattus norvegicus | ||
11. | ALA2074837 | Tetrahexylammonium | Inhibition | 0 | ALA2078186 | inhibitor [90-95 % inhibition] | % | Rattus norvegicus | ||||
12. | ALA331320 | Dimethylamiloride | Inhibition | 0 | ALA2078197 | inhibitor [90-95 % inhibition] | % | Rattus norvegicus | ||||
13. | desipramine | desmethylimipramine | Inhibition | 0 | ALA2078196 | inhibitor [90-95 % inhibition] | % | Rattus norvegicus | ||||
14. | cefluprenam | Cefluprenam | Activity | = | 76 | % | ALA2078210 | inhibitor [76 % of control] | % | Rattus norvegicus | ||
15. | Acetyl-L-Carnitine | SID11113462 | Activity | 0 | ALA2076296 | substrate [+] | Rattus norvegicus | |||||
16. | (±)-Propionylcarnitine chloride | Propionyl-Carnitine | Activity | 0 | ALA2076296 | substrate [+] | Rattus norvegicus | |||||
17. | 4-Amino-N-(2-diethylaminoethyl)benzamide | Procainamide | Inhibition | 0 | ALA2078188 | inhibitor [50-75 % inhibition] | % | Rattus norvegicus | ||||
18. | ALA3 | 2 | Inhibition | 0 | ALA2078190 | inhibitor [50-75 % inhibition] | % | Rattus norvegicus | ||||
19. | 1-Methyl-4-phenyl-1,2,3,6-tetrahydropyridine, free base | MPTP | Inhibition | 0 | ALA2078192 | inhibitor [50-75 % inhibition] | % | Rattus norvegicus | ||||
20. | MPP⁺ | 1 | Inhibition | 0 | ALA2078193 | inhibitor [50-75 % inhibition] | % | Rattus norvegicus |