# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5195146 | 10 | deltaTm | <= | 70 | degrees C | ALA5098743 | degrees C | Homo sapiens | |||
2. | ALA5174454 | 7; 14215 | deltaTm | <= | 70 | degrees C | ALA5098743 | degrees C | Homo sapiens | |||
3. | LCL161 | 3, LCL161 | deltaTm | = | 58 | degrees C | ALA5098743 | degrees C | Homo sapiens | |||
4. | ALA5174454 | 7; 14215 | Kinact | = | 1.046 | /min | ALA5098741 | /min | Homo sapiens | |||
5. | ALA5174454 | 7; 14215 | Ki | = | 0.185 | uM | ALA5098740 | 6.73 | nM | Homo sapiens | ||
6. | ALA5174454 | 7; 14215 | Activity | 0 | ALA5098737 | Active | Homo sapiens | |||||
7. | ALA5174454 | 7; 14215 | Activity | 0 | ALA5098735 | Active | Homo sapiens | |||||
8. | ALA5195146 | 10 | IC50 | = | 291 | nM | ALA5098731 | 6.54 | nM | Homo sapiens | ||
9. | ALA5174454 | 7; 14215 | IC50 | = | 11 | nM | ALA5098731 | 7.96 | nM | Homo sapiens | ||
10. | LCL161 | 3, LCL161 | IC50 | = | 15 | nM | ALA5098731 | 7.82 | nM | Homo sapiens | ||
11. | ALA5195146 | 10 | IC50 | = | 278 | nM | ALA5098727 | 6.56 | nM | Homo sapiens | ||
12. | ALA5170823 | 9 | IC50 | = | 482 | nM | ALA5098727 | 6.32 | nM | Homo sapiens | ||
13. | ALA5203019 | 8 | IC50 | = | 556 | nM | ALA5098727 | 6.25 | nM | Homo sapiens | ||
14. | ALA5174454 | 7; 14215 | IC50 | = | 43 | nM | ALA5098727 | 7.37 | nM | Homo sapiens | ||
15. | ALA5191180 | 6 | IC50 | = | 319 | nM | ALA5098727 | 6.50 | nM | Homo sapiens | ||
16. | ALA5200297 | 5 | IC50 | > | 1000 | nM | ALA5098727 | nM | Homo sapiens | |||
17. | ALA5193194 | 4 | IC50 | = | 280 | nM | ALA5098727 | 6.55 | nM | Homo sapiens | ||
18. | ALA5169527 | 3 | IC50 | = | 866 | nM | ALA5098727 | 6.06 | nM | Homo sapiens | ||
19. | ALA5175233 | 2 | IC50 | = | 50 | nM | ALA5098727 | 7.30 | nM | Homo sapiens | ||
20. | ALA5181541 | 1 | IC50 | = | 35 | nM | ALA5098727 | 7.46 | nM | Homo sapiens |