| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  [³H]taurocholic acid | THCA | Activity | 0 | ALA2075768 | is not an inhibitor [-] | Rattus norvegicus | |||||
| 2. |  Tauroursodeoxycholic Acid | 9a, tauro | Activity | 0 | ALA2075768 | is not an inhibitor [-] | Rattus norvegicus | |||||
| 3. |  Chenodeoxycholic acid | 1 | Activity | 0 | ALA2075769 | is not an inhibitor [-] | Rattus norvegicus | |||||
| 4. | [³H]taurocholic acid | THCA | Activity | 0 | ALA2075769 | is not an inhibitor [-] | Rattus norvegicus | |||||
| 5. |  ALA307649 | rifamycin B | Activity | 0 | ALA2078332 | is not an inhibitor [-] | Rattus norvegicus | |||||
| 6. |  Mitoxantrone | Mitoxantrone | Activity | 0 | ALA2078364 | is not an inducer [-] | Rattus norvegicus | |||||
| 7. |  phenobarbital | phenobarbital | Activity | 0 | ALA2078365 | is not an inducer [-] | Rattus norvegicus | |||||
| 8. |  ALA3351088 | Endotoxin | Activity | 0 | ALA2078348 | inducer [Decrease] | Rattus norvegicus | |||||
| 9. |  ALA384467 | 9 | Activity | 0 | ALA2078347 | inducer [Decrease] | Rattus norvegicus | |||||
| 10. | ALA384467 | 9 | Activity | 0 | ALA2078362 | inducer [Decrease] | Rattus norvegicus | |||||
| 11. | ALA384467 | 9 | Activity | 0 | ALA2078354 | inducer [Decrease] | Rattus norvegicus | |||||
| 12. |  Quinidine | quinidine | Km | = | 5 | uM | ALA2075766 | substrate [Km=5uM] | nM | Rattus norvegicus | ||
| 13. |  ALA1790497 | XII | Km | = | 19.1 | uM | ALA2078268 | substrate [Km=19.1uM] | nM | Rattus norvegicus | ||
| 14. |  Ursodeoxycholic acid | UDCA | Activity | = | 39 | % | ALA2078272 | inhibitor [39 % of control] | % | Rattus norvegicus | ||
| 15. |  Taurochenodeoxycholic acid | 7 | Activity | = | 33 | % | ALA2078274 | inhibitor [33 % of control] | % | Rattus norvegicus | ||
| 16. |  taurolithocholic acid-3-sulphate | 6a, tauro | Activity | = | 16 | % | ALA2078273 | inhibitor [16 % of control] | % | Rattus norvegicus | ||
| 17. |  ALA1742475 | Flezelastine | Activity | 0 | ALA2078337 | inhibitor [+] | Rattus norvegicus | |||||
| 18. |  Azelastine | Azelastine | Activity | 0 | ALA2078338 | inhibitor [+] | Rattus norvegicus | |||||
| 19. |  grepafloxacin | 1j-2 | Activity | 0 | ALA2078275 | substrate [+] | Rattus norvegicus | |||||
| 20. |  ALA2074712 | Irinotecan (CPT-11) carboxylate | Activity | 0 | ALA2078271 | substrate [+] | Rattus norvegicus |
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