| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA4538174 | EUB0000298 | Kd | = | 140 | nM | ALA5213613 | 6.85 | nM | Homo sapiens | ||
| 2. |  PF 05105679 | 8, PF-05105679 | % of control | = | 40 | % | ALA5214525 | % | Homo sapiens | |||
| 3. |  ALA4561806 | EUB0001135 | % of control | = | 42 | % | ALA5213910 | % | Homo sapiens | |||
| 4. | ALA4561806 | EUB0001135 | Kd | > | 10 | uM | ALA5213909 | nM | Homo sapiens | |||
| 5. |  ALA4513786 | ABT-546 | % of control | = | 48 | % | ALA5213821 | % | Homo sapiens | |||
| 6. | ALA4513786 | ABT-546 | Kd | > | 10 | uM | ALA5213820 | nM | Homo sapiens | |||
| 7. |  ALA4533008 | EUB0000332a | % of control | = | 31 | % | ALA5214296 | % | Homo sapiens | |||
| 8. |  CMPD101 | 2a | IC50 | = | 5.4 | nM | ALA5150325 | 8.27 | nM | Homo sapiens | ||
| 9. |  ALA4445335 | Roxyl-ZV-5J | INH | = | 10 | % | ALA4408006 | % | Homo sapiens | |||
| 10. |  ALA4455923 | 48c | INH | < | 50 | % | ALA4405389 | % | Homo sapiens | |||
| 11. |  ALA4559936 | (+/-)-6 | Activity | = | 100 | % | ALA4391364 | % | Homo sapiens | |||
| 12. |  ALA4564973 | 50 | INH | = | 93 | % | ALA4389738 | % | Homo sapiens | |||
| 13. |  ALA4555459 | 43 | INH | = | 71 | % | ALA4389261 | % | Homo sapiens | |||
| 14. |  ALA4545456 | 24 | INH | = | 0 | % | ALA4387251 | % | Homo sapiens | |||
| 15. |  Abemaciclib | ABEMACICLIB | INH | = | 0.5 | % | ALA4387251 | % | Homo sapiens | |||
| 16. |  ALA4473365 | 7c | Activity | = | 100 | % | ALA4382542 | % | Homo sapiens | |||
| 17. |  ALA4438748 | 12j | IC50 | > | 10 | uM | ALA4379342 | nM | Homo sapiens | |||
| 18. |  CDK9-IN-7 | 21e | INH | = | 3 | % | ALA4377874 | % | Homo sapiens | |||
| 19. |  ALA4877302 | 18 | IC50 | > | 10000 | nM | ALA4810441 | nM | Homo sapiens | |||
| 20. |  ALA4847703 | 16 | IC50 | > | 10000 | nM | ALA4810441 | nM | Homo sapiens |
The page will load shortly, Thanks for your patience!