# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA2402081 | 37 | INH | = | -6 | % | ALA2406528 | % | Homo sapiens | |||
2. | ALA2397315 | 31d-2 | IC50 | = | 4.8 | uM | ALA2399037 | 5.32 | nM | Homo sapiens | ||
3. | ALA2397316 | 31-f | IC50 | = | 12 | uM | ALA2399037 | 4.92 | nM | Homo sapiens | ||
4. | ALA2386917 | 8 | INH | 0 | ALA2387907 | Not Active | % | Homo sapiens | ||||
5. | Taselisib (GDC 0032) | 11l, GDC-0032 | IC50 | > | 10 | uM | ALA2388230 | nM | Homo sapiens | |||
6. | CNX-1351 | 3, CNX-1351 | IC50(app) | > | 1 | uM | ALA2317620 | nM | Homo sapiens | |||
7. | BAY-091 | EUB0001564 | % inhibition | 4.18 | % | ALA4887999 | Not Active | % | Homo sapiens | |||
8. | BI 605906 | BI605906 | % Ctrl | 97 | % | ALA4887540 | Not Active | % | Homo sapiens | |||
9. | ALA4580220 | EUB0000311 | % residual kinase activity | 103 | % | ALA4884535 | Not Active | % | Homo sapiens | |||
10. | MLI-2 | 1; MLi-2 | % Inhibition | -0.741 | % | ALA4882863 | Not Active | % | Homo sapiens | |||
11. | ALA3417525 | 69, BI665915 | % Ctrl | 103.5 | % | ALA4882092 | Not Active | % | Homo sapiens | |||
12. | BAY-885 | BAY-885; 41 | % residual kinase activity | 96 | % | ALA4881297 | Not Active | % | Homo sapiens | |||
13. | ALA3360243 | 42 | Activity | = | 87 | % | ALA3375579 | % | Homo sapiens | |||
14. | ALA3360242 | 41 | Activity | = | 80 | % | ALA3375579 | % | Homo sapiens | |||
15. | ALA3360241 | 40 | Activity | = | 87 | % | ALA3375579 | % | Homo sapiens | |||
16. | ALA3360240 | 39 | Activity | = | 94 | % | ALA3375579 | % | Homo sapiens | |||
17. | ALA3360239 | 38 | Activity | = | 98 | % | ALA3375579 | % | Homo sapiens | |||
18. | ALA3360238 | 37 | Activity | = | 88 | % | ALA3375579 | % | Homo sapiens | |||
19. | ALA3360237 | 36 | Activity | = | 85 | % | ALA3375579 | % | Homo sapiens | |||
20. | ALA3360236 | 35 | Activity | = | 96 | % | ALA3375579 | % | Homo sapiens |