# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | Canertinib (CI-1033) | 18 | Kd | = | 1100 | nM | ALA1908438 | 5.96 | nM | Homo sapiens | ||
2. | Canertinib (CI-1033) | 18 | Kd | = | 500 | nM | ALA1908437 | 6.30 | nM | Homo sapiens | ||
3. | AT7519 | 33 | Kd | > | 10000 | nM | ALA1908438 | nM | Homo sapiens | |||
4. | Sorafenib | 5 | Kd | > | 10000 | nM | ALA1908438 | nM | Homo sapiens | |||
5. | Sorafenib | 5 | Kd | > | 10000 | nM | ALA1908437 | nM | Homo sapiens | |||
6. | Nilotinib (AMN-107) | 38 | Kd | > | 10000 | nM | ALA1908438 | nM | Homo sapiens | |||
7. | Nilotinib (AMN-107) | 38 | Kd | > | 10000 | nM | ALA1908437 | nM | Homo sapiens | |||
8. | GSK690693 | 3g, GSK-690693 | Kd | > | 10000 | nM | ALA1908438 | nM | Homo sapiens | |||
9. | GSK690693 | 3g, GSK-690693 | Kd | > | 10000 | nM | ALA1908437 | nM | Homo sapiens | |||
10. | RAF265 (CHIR-265) | CHIR-265/RAF-265 | Kd | > | 10000 | nM | ALA1908438 | nM | Homo sapiens | |||
11. | RAF265 (CHIR-265) | CHIR-265/RAF-265 | Kd | > | 10000 | nM | ALA1908437 | nM | Homo sapiens | |||
12. | AT7519 | 33 | Kd | > | 10000 | nM | ALA1908437 | nM | Homo sapiens | |||
13. | Bosutinib Isomer 1, Free Base | 1 (SKI-606) | Kd | = | 830 | nM | ALA1908438 | 6.08 | nM | Homo sapiens | ||
14. | Bosutinib Isomer 1, Free Base | 1 (SKI-606) | Kd | = | 500 | nM | ALA1908437 | 6.30 | nM | Homo sapiens | ||
15. | MLN8054 | MLN-8054 | Kd | > | 10000 | nM | ALA1908438 | nM | Homo sapiens | |||
16. | MLN8054 | MLN-8054 | Kd | > | 10000 | nM | ALA1908437 | nM | Homo sapiens | |||
17. | GSK461364 | GSK-461364A | Kd | > | 10000 | nM | ALA1908438 | nM | Homo sapiens | |||
18. | GSK461364 | GSK-461364A | Kd | > | 10000 | nM | ALA1908437 | nM | Homo sapiens | |||
19. | AST-487 (NVP-AST487) | AST-487 | Kd | = | 4400 | nM | ALA1908438 | 5.36 | nM | Homo sapiens | ||
20. | AST-487 (NVP-AST487) | AST-487 | Kd | = | 950 | nM | ALA1908437 | 6.02 | nM | Homo sapiens |