# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | pyrotinib | PYROTINIB | IC50 | = | 1836.96 | nM | ALA5162346 | 5.74 | nM | Homo sapiens | ||
2. | Neratinib (HKI-272) | 25o (table 3) | IC50 | = | 694.11 | nM | ALA5162346 | 6.16 | nM | Homo sapiens | ||
3. | ALA5178703 | 17 | IC50 | = | 6065.38 | nM | ALA5162346 | 5.22 | nM | Homo sapiens | ||
4. | ALA5182870 | 24g | IC50 | = | 8.02 | uM | ALA5156381 | 5.10 | nM | Homo sapiens | ||
5. | Tucidinostat (Chidamide) | CS055, Epidaza | IC50 | > | 10 | uM | ALA5156381 | nM | Homo sapiens | |||
6. | ALA4068334 | 16o | GI50 | = | 0.008 | uM | ALA3993299 | nM | Homo sapiens | |||
7. | ALA4760646 | 12 | CI | = | 0.43 | ALA4738174 | Homo sapiens | |||||
8. | ALA4760646 | 12 | CI | = | 0.89 | ALA4738173 | Homo sapiens | |||||
9. | ALA4760646 | 12 | CI | = | 0.87 | ALA4738172 | Homo sapiens | |||||
10. | ALA4760646 | 12 | IC50 | = | 20.73 | uM | ALA4738156 | 4.68 | nM | Homo sapiens | ||
11. | ALA4856177 | 37d | IC50 | = | 132 | nM | ALA4830451 | 6.88 | nM | Homo sapiens | ||
12. | Rucaparib | 63, AG-014699 | IC50 | = | 343.894 | uM | ALA2363848 | nM | Homo sapiens | |||
13. | CCT 018159 | 3a CCT018159 | IC50 | = | 14.787 | uM | ALA2363848 | 4.83 | nM | Homo sapiens | ||
14. | TW-37 | 5, TW-37 | IC50 | = | 3.307 | uM | ALA2363848 | 5.48 | nM | Homo sapiens | ||
15. | JNJ-26854165 (Serdemetan) | SID137276015 | IC50 | = | 27.557 | uM | ALA2363848 | 4.56 | nM | Homo sapiens | ||
16. | PF-4708671 | SID137275978 | IC50 | = | 154.149 | uM | ALA2363848 | nM | Homo sapiens | |||
17. | Avagacestat | 80 BMS-708163 | IC50 | = | 491.324 | uM | ALA2363848 | nM | Homo sapiens | |||
18. | EHT 1864 | SID137275837 | IC50 | = | 123.111 | uM | ALA2363848 | nM | Homo sapiens | |||
19. | CCT007093 | A17 | IC50 | = | 161.601 | uM | ALA2363848 | nM | Homo sapiens | |||
20. | AZD6482 | AZD-6482 | IC50 | = | 398.13 | uM | ALA2363848 | nM | Homo sapiens |