# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5266562 | 43 | Activity | 0 | ALA5237576 | Active | Homo sapiens | |||||
2. | ALA5291038 | 95; MS645 | IC50 | = | 15 | nM | ALA5227295 | 7.82 | nM | Homo sapiens | ||
3. | ALA2326284 | 17 | EC50 | = | 1.2 | uM | ALA5227273 | 5.92 | nM | Homo sapiens | ||
4. | EPZ015666 | 1; EPZ015666 | IC50 | = | 5 | uM | ALA5227254 | 5.30 | nM | Homo sapiens | ||
5. | Palbociclib | 43(table 3) | EC50 | = | 1.4 | uM | ALA5227244 | 5.85 | nM | Homo sapiens | ||
6. | ALA5196874 | (-)-53; MU1656 | Activity | 0 | ALA5161971 | NA | Homo sapiens | |||||
7. | Dinaciclib (SCH727965) | DINACICLIB | FC | = | 2.5 | ALA4775155 | Homo sapiens | |||||
8. | ALA492323 | 2 | INH | 0 | ALA4338031 | Active | % | Homo sapiens | ||||
9. | ALA492323 | 2 | INH | 0 | ALA4338030 | Active | % | Homo sapiens | ||||
10. | ALA492323 | 2 | Activity | 0 | ALA4337993 | Dose-dependent effect | Homo sapiens | |||||
11. | ALA492323 | 2 | INH | 0 | ALA4337995 | Active | % | Homo sapiens | ||||
12. | ALA492323 | 2 | INH | 0 | ALA4337997 | Active | % | Homo sapiens | ||||
13. | ALA492323 | 2 | Activity | 0 | ALA4337999 | Active | Homo sapiens | |||||
14. | ALA492323 | 2 | Activity | 0 | ALA4338001 | Active | Homo sapiens | |||||
15. | ALA492323 | 2 | Activity | 0 | ALA4338007 | Dose-dependent effect | Homo sapiens | |||||
16. | ALA492323 | 2 | Activity | 0 | ALA4338021 | Active | Homo sapiens | |||||
17. | ALA492323 | 2 | INH | 0 | ALA4338027 | Dose-dependent effect | % | Homo sapiens | ||||
18. | ALA492323 | 2 | INH | 0 | ALA4338026 | Dose-dependent effect | % | Homo sapiens | ||||
19. | ALA492323 | 2 | INH | 0 | ALA4338025 | Dose-dependent effect | % | Homo sapiens | ||||
20. | ALA4292680 | 3 | Activity | >= | 15 | % | ALA4251866 | % | Homo sapiens |