# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | AG-270 | 153 | INH | = | 81.1 | % | ALA4835592 | % | Homo sapiens | |||
2. | AG-270 | 153 | INH | = | 63.5 | % | ALA4835591 | % | Homo sapiens | |||
3. | AG-270 | 153 | INH | = | 44.7 | % | ALA4835590 | % | Homo sapiens | |||
4. | AG-270 | 153 | INH | = | 33.4 | % | ALA4835589 | % | Homo sapiens | |||
5. | AG-270 | 153 | TGI | = | 67 | % | ALA4835588 | % | Homo sapiens | |||
6. | AG-270 | 153 | TGI | = | 66 | % | ALA4835587 | % | Homo sapiens | |||
7. | AG-270 | 153 | TGI | = | 48 | % | ALA4835586 | % | Homo sapiens | |||
8. | AG-270 | 153 | TGI | = | 36 | % | ALA4835585 | % | Homo sapiens | |||
9. | ALA4281829 | 13a | Activity | 0 | ALA4269288 | Non-Toxic | Homo sapiens | |||||
10. | ALA4281829 | 13a | Activity | 0 | ALA4269286 | Non-Toxic | Homo sapiens | |||||
11. | ALA4281829 | 13a | Activity | 0 | ALA4269284 | Active | Homo sapiens | |||||
12. | Lopinavir | 1a, ABT-378 Lopinavir | Activity | 0 | ALA4269284 | Not Active | Homo sapiens | |||||
13. | ALA4281829 | 13a | Activity | 0 | ALA4269283 | Non-Toxic | Homo sapiens | |||||
14. | ALA5268484 | 11; GNE-375 | IC50 | = | 2 | uM | ALA5262013 | 5.70 | nM | Homo sapiens | ||
15. | ALA5270178 | 5 | IC50 | = | 20 | uM | ALA5262013 | 4.70 | nM | Homo sapiens | ||
16. | ALA5282240 | 3 | IC50 | = | 20 | uM | ALA5262013 | 4.70 | nM | Homo sapiens | ||
17. | Rucaparib | 63, AG-014699 | IC50 | = | 21.434 | uM | ALA2363345 | 4.67 | nM | Homo sapiens | ||
18. | CCT 018159 | 3a CCT018159 | IC50 | = | 69.558 | uM | ALA2363345 | 4.16 | nM | Homo sapiens | ||
19. | TW-37 | 5, TW-37 | IC50 | = | 0.455 | uM | ALA2363345 | 6.34 | nM | Homo sapiens | ||
20. | JNJ-26854165 (Serdemetan) | SID137276015 | IC50 | = | 10.183 | uM | ALA2363345 | 4.99 | nM | Homo sapiens |