# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | pyrotinib | PYROTINIB | IC50 | = | 1559.06 | nM | ALA5162344 | 5.81 | nM | Homo sapiens | ||
2. | Neratinib (HKI-272) | 25o (table 3) | IC50 | = | 1291.95 | nM | ALA5162344 | 5.89 | nM | Homo sapiens | ||
3. | ALA5178703 | 17 | IC50 | = | 3967.21 | nM | ALA5162344 | 5.40 | nM | Homo sapiens | ||
4. | Rucaparib | 63, AG-014699 | IC50 | = | 332.401 | uM | ALA2363418 | nM | Homo sapiens | |||
5. | CCT 018159 | 3a CCT018159 | IC50 | = | 591.959 | uM | ALA2363418 | nM | Homo sapiens | |||
6. | TW-37 | 5, TW-37 | IC50 | = | 4.588 | uM | ALA2363418 | 5.34 | nM | Homo sapiens | ||
7. | JNJ-26854165 (Serdemetan) | SID137276015 | IC50 | = | 176.439 | uM | ALA2363418 | nM | Homo sapiens | |||
8. | PF-4708671 | SID137275978 | IC50 | = | 252.746 | uM | ALA2363418 | nM | Homo sapiens | |||
9. | Avagacestat | 80 BMS-708163 | IC50 | = | 555.911 | uM | ALA2363418 | nM | Homo sapiens | |||
10. | EHT 1864 | SID137275837 | IC50 | = | 1082.431 | uM | ALA2363418 | nM | Homo sapiens | |||
11. | CCT007093 | A17 | IC50 | = | 505.947 | uM | ALA2363418 | nM | Homo sapiens | |||
12. | AZD6482 | AZD-6482 | IC50 | = | 103.832 | uM | ALA2363418 | nM | Homo sapiens | |||
13. | ALA1614701 | AZD-6244 | IC50 | = | 69.025 | uM | ALA2363418 | 4.16 | nM | Homo sapiens | ||
14. | SB590885 | 33, SB-590885 | IC50 | = | 358.916 | uM | ALA2363418 | nM | Homo sapiens | |||
15. | PD0325901 | 34, PD-0325901 | IC50 | = | 11.633 | uM | ALA2363418 | 4.93 | nM | Homo sapiens | ||
16. | AZD8055 | 10, AZD-8055 | IC50 | = | 0.43 | uM | ALA2363418 | 6.37 | nM | Homo sapiens | ||
17. | GDC-0941 | 17, GDC-0941 | IC50 | = | 0.418 | uM | ALA2363418 | 6.38 | nM | Homo sapiens | ||
18. | BEZ235 | SID124898663 | IC50 | = | 0.01 | uM | ALA2363418 | 8.00 | nM | Homo sapiens | ||
19. | Palbociclib | 43(table 3) | IC50 | = | 212.067 | uM | ALA2363418 | nM | Homo sapiens | |||
20. | MK-2206 | 17 | IC50 | = | 0.965 | uM | ALA2363418 | 6.02 | nM | Homo sapiens |