# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5267741 | 2 | Activity | 0 | ALA5230033 | Not Active | Homo sapiens | |||||
2. | ALA5286325 | 1 | Activity | 0 | ALA5230033 | Active | Homo sapiens | |||||
3. | ALA5196874 | (-)-53; MU1656 | Activity | 0 | ALA5162033 | NA | Homo sapiens | |||||
4. | Rucaparib | 63, AG-014699 | IC50 | = | 102.833 | uM | ALA2363598 | nM | Homo sapiens | |||
5. | CCT 018159 | 3a CCT018159 | IC50 | = | 6.593 | uM | ALA2363598 | 5.18 | nM | Homo sapiens | ||
6. | TW-37 | 5, TW-37 | IC50 | = | 0.035 | uM | ALA2363598 | 7.45 | nM | Homo sapiens | ||
7. | JNJ-26854165 (Serdemetan) | SID137276015 | IC50 | = | 8.823 | uM | ALA2363598 | 5.05 | nM | Homo sapiens | ||
8. | PF-4708671 | SID137275978 | IC50 | = | 32.675 | uM | ALA2363598 | 4.49 | nM | Homo sapiens | ||
9. | Avagacestat | 80 BMS-708163 | IC50 | = | 26.878 | uM | ALA2363598 | 4.57 | nM | Homo sapiens | ||
10. | EHT 1864 | SID137275837 | IC50 | = | 95.606 | uM | ALA2363598 | 4.02 | nM | Homo sapiens | ||
11. | CCT007093 | A17 | IC50 | = | 143.397 | uM | ALA2363598 | nM | Homo sapiens | |||
12. | AZD6482 | AZD-6482 | IC50 | = | 4.344 | uM | ALA2363598 | 5.36 | nM | Homo sapiens | ||
13. | ALA1614701 | AZD-6244 | IC50 | = | 34.032 | uM | ALA2363598 | 4.47 | nM | Homo sapiens | ||
14. | SB590885 | 33, SB-590885 | IC50 | = | 536.593 | uM | ALA2363598 | nM | Homo sapiens | |||
15. | PD0325901 | 34, PD-0325901 | IC50 | = | 0.454 | uM | ALA2363598 | 6.34 | nM | Homo sapiens | ||
16. | AZD8055 | 10, AZD-8055 | IC50 | = | 3.965 | uM | ALA2363598 | 5.40 | nM | Homo sapiens | ||
17. | GDC-0941 | 17, GDC-0941 | IC50 | = | 8.349 | uM | ALA2363598 | 5.08 | nM | Homo sapiens | ||
18. | BEZ235 | SID124898663 | IC50 | = | 0.124 | uM | ALA2363598 | 6.91 | nM | Homo sapiens | ||
19. | Palbociclib | 43(table 3) | IC50 | = | 32.823 | uM | ALA2363598 | 4.48 | nM | Homo sapiens | ||
20. | MK-2206 | 17 | IC50 | = | 276.007 | uM | ALA2363598 | nM | Homo sapiens |